SCHEMBL7969434

SCHEMBL7969434

Cc1cc(C(C)(C)C)ccc1CC#N

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1D P28221 2/20 0.43
ADRA2A P08913 1/20 0.43
ADRA2B P18089 1/20 0.43
ADRA2C P18825 1/20 0.43
ADRA1D P25100 1/20 0.43
HTR1B P28222 1/20 0.43
ADRA1A P35348 1/20 0.43
ADRA1B P35368 1/20 0.43
CYP1A2 P05177 2/20 0.42
CYP2C19 P33261 2/20 0.42
EPHX2 P34913 1/20 0.38
RXRA P19793 1/20 0.37
RXRB P28702 1/20 0.37
KIF11 P52732 1/20 0.37
TSHR P16473 2/20 0.37
KDM4E B2RXH2 2/20 0.37
ALDH1A1 P00352 4/20 0.36
HPGD P15428 2/20 0.36
ALOX15 P16050 1/20 0.36
HSD17B10 Q99714 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25786471 0.83 DAO (0.43) RXRARXRBKIF11MAPTPOLB
SCHEMBL7918774 0.81 CYP1A2 (0.40) HTR1DCYP1A2CYP2C19RXRARXRB
SCHEMBL29284733 0.81 CYP1A2 (0.40) HTR1DADRA2AADRA2BADRA2CADRA1D
SCHEMBL1822997 0.78 PYCR1 (0.44) TSHRKDM4EALDH1A1HPGDALOX15
SCHEMBL10835974 0.78 MAPT (0.37) HTR1DADRA2AADRA2BADRA2CADRA1D
SCHEMBL195863 0.75 CASP1 (0.44) KDM4EALDH1A1HSD17B10CYP2D6L3MBTL1
SCHEMBL1773826 0.75 TDO2 (0.40) CYP2C19RXRARXRBKIF11TSHR
SCHEMBL5651750 0.74 ALDH1A1 (0.46) TSHRKDM4EALDH1A1ALOX15L3MBTL1
SCHEMBL1096617 0.74 CYP2A6 (0.49) CYP1A2CYP2C19KDM4ETDP1L3MBTL1
SCHEMBL5786 0.74 CSNK2A1 (0.49) TSHRALDH1A1L3MBTL1LMNAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6288101-B1 ADMINISTERING COMPOUNDS SUCH AS 2,6-DIMETHYL-4-ISOPROPYLBENZALDEHYDE TO TREAT INDICATIONS WHERE STIMULATION OF SUBTYPES OF THE SEROTONIN RECEPTOR IS IMPLICATED, SUCH AS MIGRAINES VIRGINIA COMMONWEALTH UNIVERSITY 2001-09-11 US disclosed
US-6124338-A TREATING MIGRAINE HEADACHE VIRGINIA COMMONWEALTH UNIVERSITY (US) 2000-09-26 US disclosed
US-6048862-A Benzylamidine derivatives with serotonin receptor binding activity VIRGINIA COMMONWEALTH UNIVERSITY (US) 2000-04-11 US disclosed
US-5969137-A TREATMENT OF NERVOUS SYSTEM DISORDERS VIRGINIA COMMONWEALTH UNIVERSITY (US) 1999-10-19 US disclosed
WO-1998012183-A1 IMIDAZOLES WITH SEROTONIN RECEPTOR BINDING ACTIVITY ALLELIX BIOPHARMACEUTICALS INC. (CA) 1998-03-26 WO disclosed