SCHEMBL7971730

SCHEMBL7971730

Cc1ccc(CC(c2cnc[nH]2)N2C(=O)COc3c(C(=O)O)cccc32)cc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CPA1 P15085 1/20 0.37
CPB2 Q96IY4 6/20 0.34
TP53 P04637 1/20 0.33
POLB P06746 1/20 0.33
HIF1A Q16665 1/20 0.32
ALDH1A1 P00352 1/20 0.32
GAA P10253 1/20 0.32
KMT2A Q03164 1/20 0.32
CYP19A1 P11511 1/20 0.32
CPB1 P15086 2/20 0.32
HTR1A P08908 1/20 0.31
HTR1D P28221 1/20 0.31
HTR1B P28222 1/20 0.31
SLC6A4 P31645 1/20 0.31
KCNH2 Q12809 1/20 0.31
XIAP P98170 1/20 0.30
BRS3 P32247 1/20 0.30
FABP4 P15090 1/20 0.30
ALOX5 P09917 1/20 0.30
PTGS2 P35354 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7967524 0.91 CPA1 (0.37) CPA1CPB2HIF1AKMT2ACPB1
SCHEMBL7971542 0.91 CPA1 (0.39) CPA1CPB2HIF1AALDH1A1KMT2A
SCHEMBL7971636 0.83 CPA1 (0.38) CPA1CPB2TP53CYP19A1CPB1
SCHEMBL7974145 0.78 CPA1 (0.36) CPA1CPB2CYP19A1CPB1BRS3
SCHEMBL7968421 0.74 CPA1 (0.40) CPA1CPB2ALDH1A1CPB1
SCHEMBL7971099 0.74 CPA1 (0.38) CPA1CPB2CPB1BRS3
SCHEMBL7971115 0.71 CPA1 (0.36) CPA1CPB2CPB1
SCHEMBL7972160 0.70 ITGA4 (0.38) ALDH1A1KMT2A
SCHEMBL7971733 0.69 KMT2A (0.41) TP53POLBALDH1A1GAAKMT2A
SCHEMBL7969211 0.66 CPA1 (0.42) CPA1CPB2ALDH1A1CYP19A1CPB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001009127-A1 BENZOXAZINE DERIVATIVES AND THEIR THERAPEUTIC USE AVENTIS PHARMA S.A. (FR) 2001-02-08 WO disclosed