SCHEMBL7972441

SCHEMBL7972441

CC(C)C(C#N)(CCCCl)c1ccccc1F

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.51
EBP Q15125 2/20 0.40
SIGMAR1 Q99720 2/20 0.40
CYP3A4 P08684 5/20 0.34
ABCB1 P08183 5/20 0.32
CYP3A5 P20815 1/20 0.31
ABCC1 P33527 3/20 0.30
CYP2C19 P33261 2/20 0.30
MEN1 O00255 1/20 0.30
SLC22A1 O15245 1/20 0.30
CACNA1F O60840 1/20 0.30
ABCB11 O95342 1/20 0.30
CHRM2 P08172 1/20 0.30
HTR1A P08908 1/20 0.30
ADRA2A P08913 1/20 0.30
CYP2C8 P10632 1/20 0.30
CYP2D6 P10635 1/20 0.30
DRD2 P14416 1/20 0.30
ADRA2B P18089 1/20 0.30
ADRA2C P18825 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7968378 0.84 L3MBTL1 (0.40) L3MBTL1EBPSIGMAR1CYP3A4ABCB1
SCHEMBL5236598 0.79 EBP (0.59) L3MBTL1EBPSIGMAR1CYP3A4ABCB1
SCHEMBL5753392 0.79 L3MBTL1 (0.44) L3MBTL1EBPSIGMAR1CYP3A4
SCHEMBL7966884 0.78 EBP (0.47) L3MBTL1EBPSIGMAR1CYP3A4ABCB1
SCHEMBL7129611 0.78 L3MBTL1 (0.43) L3MBTL1EBPSIGMAR1CYP2C19MEN1
SCHEMBL7956602 0.77 SIGMAR1 (0.58) L3MBTL1EBPSIGMAR1CYP3A4ABCB1
SCHEMBL7956311 0.77 EBP (0.46) L3MBTL1EBPSIGMAR1CYP3A4ABCB1
SCHEMBL5227349 0.77 L3MBTL1 (0.44) L3MBTL1EBPSIGMAR1MEN1CHRM2
SCHEMBL7956207 0.76 SIGMAR1 (0.48) L3MBTL1EBPSIGMAR1CYP3A4ABCB1
SCHEMBL7956313 0.76 SIGMAR1 (0.73) L3MBTL1EBPSIGMAR1CYP3A4ABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265439-B1 Halogenated phenylacetonitrile alkylaminoalkylphenyl compounds as immunosuppressives G.D. SEARLE & CO. 2001-07-24 US disclosed
US-5451604-A Useful in organ transplant surgery G. D. SEARLE & CO. (US) 1995-09-19 US disclosed