SCHEMBL7974196

SCHEMBL7974196

NC(=O)c1ccc2nc(C3=NCC(c4cccc(Br)c4)=C3O)[nH]c2c1

nearest known ligand 0.55

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CHEK2 O96017 18/20 0.55
HDAC3 O15379 1/20 0.54
HDAC1 Q13547 1/20 0.54
HDAC2 Q92769 1/20 0.54
HDAC8 Q9BY41 1/20 0.54
HDAC6 Q9UBN7 1/20 0.54
PKN1 Q16512 1/20 0.48
PKN2 Q16513 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7982194 0.81 NPC1 (0.52) HDAC3HDAC1HDAC2HDAC8HDAC6
SCHEMBL10139807 0.75 F9 (0.56) CHEK2HDAC3HDAC1HDAC2HDAC8
SCHEMBL10140086 0.74 PLAU (0.67) CHEK2
SCHEMBL7972153 0.74 CHEK2 (0.54) CHEK2HDAC3HDAC1HDAC2HDAC8
SCHEMBL2341761 0.73 HDAC6 (0.77) CHEK2HDAC3HDAC1HDAC2HDAC8
SCHEMBL2649653 0.72 HDAC6 (0.76) CHEK2HDAC3HDAC1HDAC2HDAC8
SCHEMBL18229615 0.71 HDAC6 (1.00) HDAC3HDAC1HDAC2HDAC8HDAC6
SCHEMBL20982670 0.70 CHEK2 (0.86) CHEK2PKN1PKN2
SCHEMBL6260767 0.70 MMP2 (0.78) CHEK2HDAC6PKN1PKN2
SCHEMBL10140770 0.70 CHEK2 (0.51) CHEK2HDAC3HDAC1HDAC2HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009143039-A2 HETEROCYCLIC COMPOUNDS AS FACTOR IXA INHIBITORS SCHERING CORPORATION (US) 2009-11-26 WO disclosed