SCHEMBL7975660

SCHEMBL7975660

CN1[C@@H]2CC[C@H]1CC(c1c(Cl)c(Cl)c(C3C[C@H]4CC[C@@H](C3)N4C)c(C(=O)O)c1C(=O)O)C2

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 4/20 0.39
HTR3E A5X5Y0 2/20 0.39
HTR3B O95264 2/20 0.39
HTR3A P46098 2/20 0.39
HTR3D Q70Z44 2/20 0.39
HTR3C Q8WXA8 2/20 0.39
HSD17B10 Q99714 2/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
CYP1A2 P05177 2/20 0.39
GMNN O75496 1/20 0.39
ALOX15 P16050 1/20 0.39
TSHR P16473 1/20 0.39
MTOR P42345 1/20 0.39
PMP22 Q01453 1/20 0.39
LMNA P02545 3/20 0.38
CYP2C19 P33261 2/20 0.38
GAA P10253 1/20 0.38
CYP2C9 P11712 2/20 0.38
CHRNA7 P36544 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7975657 1.00 CYP2D6 (0.39) CYP2D6HTR3EHTR3BHTR3AHTR3D
SCHEMBL7973796 0.74 HTR3E (0.40) CYP2D6HTR3EHTR3BHTR3AHTR3D
SCHEMBL7973793 0.74 HTR3E (0.40) CYP2D6HTR3EHTR3BHTR3AHTR3D
SCHEMBL7265701 0.73 HTR3A (0.49) CYP2D6HTR3EHTR3BHTR3AHTR3D
SCHEMBL6139012 0.73 HTR3A (0.49) CYP2D6HTR3EHTR3BHTR3AHTR3D
SCHEMBL9472450 0.73 HTR3A (0.49) CYP2D6HTR3EHTR3BHTR3AHTR3D
SCHEMBL9871559 0.73 HTR3A (0.49) CYP2D6HTR3EHTR3BHTR3AHTR3D
SCHEMBL7484945 0.68 HTR3A (0.47) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL7267112 0.68 HTR3E (0.45) CYP2D6HTR3EHTR3BHTR3AHTR3D
SCHEMBL7273067 0.68 HTR3E (0.45) CYP2D6HTR3EHTR3BHTR3AHTR3D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6274623-B1 DI- OR POLY-ALKOXY-OR ACYLOXY-SUBSTITUTED ARALKYL AND ARAKENYL QUATERNARY AMMONIUM DERIVATIVES OF CYCLIC AMINOALKANOL DIESTERS SUCH AS BIS(N-(3,4-DIPROPIONYLOXY-BENZYL)GRANATANINIUM-3-ALPHA-YL)ADIPATE DIBROMIDE NEWLAXANT LLC 2001-08-14 US disclosed
US-5990124-A ALKOXY AND/OR ACYLOXY DI- AND POLY-SUBSTITUTED ARALKYL AND ARALKENYL BIS-QUATERNARY AMMONIUM DERIVATIVES OF CYCLIC ALKANOL DIESTERS; SUCH AS BIS(N-(4-ACETOXY-3-METHOXYBENZYL) TROPANIUM-3-YL)-3,6-ENDOMETHYLENE-1,2,3,6-TETRAHYDROPHTHALATE GYERMEK LASZLO (US) 1999-11-23 US disclosed