SCHEMBL7484945

SCHEMBL7484945

CN1C2CCC1CC(c1c(C(=O)O)c3ccccc3n(C)c1=O)C2

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 11/20 0.47
HTR3E A5X5Y0 5/20 0.47
HTR3B O95264 5/20 0.47
HTR3D Q70Z44 5/20 0.47
HTR3C Q8WXA8 5/20 0.47
EGFR P00533 1/20 0.46
ALDH1A1 P00352 2/20 0.45
KDM4E B2RXH2 1/20 0.45
GAA P10253 1/20 0.45
HPGD P15428 1/20 0.45
HSD17B10 Q99714 1/20 0.45
PADI4 Q9UM07 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7443724 0.87 HTR3A (0.50) HTR3AHTR3EHTR3BHTR3DHTR3C
SCHEMBL7434788 0.85 HTR3A (0.52) HTR3AHTR3EHTR3BHTR3DHTR3C
SCHEMBL7432574 0.83 HTR3A (0.60) HTR3AHTR3EHTR3BHTR3DHTR3C
SCHEMBL7430512 0.82 HTR3E (0.56) HTR3AHTR3EHTR3BHTR3DHTR3C
SCHEMBL7444191 0.76 HTR3E (0.45) HTR3AHTR3EHTR3BHTR3DHTR3C
SCHEMBL7430595 0.73 HTR3A (0.67) HTR3AHTR3EHTR3BHTR3DHTR3C
SCHEMBL7437202 0.71 ALDH1A1 (0.62) EGFRALDH1A1KDM4EGAAHPGD
SCHEMBL6672250 0.70 HTR3E (0.50) HTR3AHTR3EHTR3BHTR3DHTR3C
SCHEMBL29701 0.70 ALDH1A1 (0.59) EGFRALDH1A1KDM4E
SCHEMBL984736 0.69 EGFR (0.65) EGFRALDH1A1KDM4EGAAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5248684-A CERTAIN 2-OXO-QUINOLINE CARBOXYLATES OR CORRESPONDING CARBOXAMIDES USEFUL AS ANTI-EMETICS AND SUPPRESSANTS OF MIGRAINE KYOWA HAKKO KOGYO CO., LTD. (JP) 1993-09-28 US disclosed
EP-0458636-A1 Antiemetic and migraine suppressing heterocyclic compounds and pharmaceutical compositions containing them KYOWA HAKKO KOGYO CO., LTD (JP) 1991-11-27 EP disclosed