SCHEMBL7977170

SCHEMBL7977170

[NH]C(=O)CCC(=O)c1ccncc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTNNB1 P35222 2/20 0.54
WNT3A P56704 2/20 0.54
PLOD2 O00469 2/20 0.52
PLOD3 O60568 2/20 0.52
PLOD1 Q02809 2/20 0.52
CYP1A2 P05177 2/20 0.52
CYP3A4 P08684 2/20 0.52
CYP2D6 P10635 2/20 0.52
CYP2C19 P33261 2/20 0.52
ALDH1A1 P00352 2/20 0.52
CYP2C9 P11712 1/20 0.52
HPGD P15428 1/20 0.52
HIF1A Q16665 1/20 0.52
NAPRT Q6XQN6 1/20 0.46
MMP1 P03956 1/20 0.46
KDM4E B2RXH2 2/20 0.45
MPO P05164 1/20 0.45
ADORA3 P0DMS8 1/20 0.45
CYP2A6 P11509 1/20 0.45
KMT2A Q03164 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15988710 0.89 CYP2C19 (0.61) CTNNB1WNT3APLOD2PLOD3PLOD1
SCHEMBL10843960 0.81 NR4A2 (0.65) CTNNB1WNT3APLOD2PLOD3PLOD1
SCHEMBL9195700 0.81 ALDH1A1 (0.77) CTNNB1WNT3APLOD2PLOD3PLOD1
SCHEMBL7977172 0.79 CYP1A2 (0.52) CTNNB1WNT3APLOD2PLOD3PLOD1
SCHEMBL31561725 0.78 ALDH1A1 (0.59) CTNNB1WNT3APLOD2PLOD3PLOD1
Propyl 4-Pyridyl Ketone SCHEMBL4952700 0.77 HSD17B3 (0.61) CTNNB1WNT3APLOD2PLOD3PLOD1
SCHEMBL7265428 0.77 PLOD2 (0.53) CTNNB1WNT3APLOD2PLOD3PLOD1
SCHEMBL16404441 0.77 CYP1A2 (0.59) CTNNB1WNT3APLOD2PLOD3PLOD1
SCHEMBL7387908 0.76 MMP1 (0.73) PLOD2PLOD3PLOD1CYP1A2CYP3A4
SCHEMBL10948430 0.75 PLOD2 (0.83) PLOD2PLOD3PLOD1CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001007409-A1 CARBAZOLE DERIVATIVES AND THEIR USE AS NEUROPEPTIDE Y5 RECEPTOR LIGANDS ASTRAZENECA UK LIMITED (GB) 2001-02-01 WO disclosed