SCHEMBL7977314

SCHEMBL7977314

O=S(=O)(Cl)c1sc(Cc2ccc3c(c2)OCO3)c(S(=O)(=O)Cl)c1-c1ccsc1Cc1ccc2c(c1)OCO2

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.39
HSD17B10 Q99714 2/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
EDNRB P24530 2/20 0.37
EDNRA P25101 2/20 0.37
MAPK8 P45983 1/20 0.36
MAPT P10636 5/20 0.36
HPGD P15428 5/20 0.36
KDM4E B2RXH2 3/20 0.36
LMNA P02545 3/20 0.36
SMN1; SMN2 Q16637 3/20 0.36
HTT P42858 1/20 0.36
POLB P06746 2/20 0.35
ATM Q13315 1/20 0.35
RAB9A P51151 2/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
GAA P10253 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7339955 0.77 EDNRA (0.45) ALDH1A1HSD17B10L3MBTL1EDNRBEDNRA
SCHEMBL6958979 0.77 EDNRA (0.45) ALDH1A1HSD17B10L3MBTL1EDNRBEDNRA
SCHEMBL6956724 0.73 ALDH1A1 (0.43) ALDH1A1HSD17B10L3MBTL1MAPTHPGD
SCHEMBL108697 0.70 ALDH1A1 (0.51) ALDH1A1HSD17B10MAPT
SCHEMBL4631437 0.69 EDNRA (0.57) EDNRBEDNRAMAPK8POLB
SCHEMBL4631407 0.68 RORB (0.50) ALDH1A1HSD17B10MAPTHPGDSMN1; SMN2
SCHEMBL7404511 0.68 RORB (0.50) ALDH1A1HSD17B10MAPTHPGDSMN1; SMN2
SCHEMBL8445530 0.64 ALDH1A1 (0.46) ALDH1A1HSD17B10L3MBTL1MAPTHPGD
SCHEMBL109195 0.63 TAAR1 (0.64) ALDH1A1MAPTGAA
SCHEMBL108235 0.62 TAAR1 (0.55) ALDH1A1HSD17B10MAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6331637-B1 N-Alkyl, N-Alkenyl, N-Alkynyl, N-Aryl and N-fused bicyclo or tricyclo thienyl-, furyl-,and Pyrrolyl-sulfonamides and derivatives thereof that modulate the activity of endothelin TEXAS BIOTECHNOLOGY CORPORATION 2001-12-18 US disclosed