SCHEMBL7980229

SCHEMBL7980229

O=C(CCl)N(c1ccccc1)c1ccccn1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 6/20 0.66
RAB9A P51151 6/20 0.66
ALDH1A1 P00352 5/20 0.66
KMT2A Q03164 4/20 0.66
NPSR1 Q6W5P4 4/20 0.66
HTT P42858 3/20 0.66
POLB P06746 2/20 0.66
MEN1 O00255 3/20 0.47
MITF O75030 2/20 0.47
TDP1 Q9NUW8 1/20 0.47
PTGIR P43119 1/20 0.46
PAX8 Q06710 4/20 0.45
SMN1; SMN2 Q16637 3/20 0.45
TP53 P04637 2/20 0.45
GLA P06280 1/20 0.45
LMNA P02545 1/20 0.45
TSHR P16473 1/20 0.43
MAPT P10636 2/20 0.43
KDM4E B2RXH2 2/20 0.43
HKDC1 Q2TB90 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7981944 0.84 PTGIR (0.46) NPC1RAB9AALDH1A1KMT2ANPSR1
SCHEMBL7982394 0.84 PTGIR (0.46) NPC1RAB9AALDH1A1KMT2ANPSR1
SCHEMBL28682606 0.81 PTGIR (0.44) NPC1RAB9AALDH1A1KMT2ANPSR1
SCHEMBL7978941 0.81 TP53 (0.51) NPC1RAB9AALDH1A1KMT2ANPSR1
SCHEMBL10855054 0.81 NPSR1 (0.50) NPC1RAB9AALDH1A1KMT2ANPSR1
SCHEMBL2345303 0.80 ALDH1A1 (1.00) NPC1RAB9AALDH1A1KMT2ANPSR1
SCHEMBL7981765 0.80 PTGIR (0.49) KMT2ANPSR1HTTPOLBMEN1
SCHEMBL10668533 0.80 NPSR1 (0.63) NPC1RAB9AALDH1A1KMT2ANPSR1
SCHEMBL7980404 0.79 LTB4R2 (0.43) KMT2ANPSR1HTTPOLBMEN1
SCHEMBL3475461 0.78 NPSR1 (0.47) NPC1RAB9AALDH1A1KMT2ANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6235730-B1 ANTICHOLESTEROL AGENT, ANTILIPEMIC AGENT JAPAN TOBACCO, INC. (JP) 2001-05-22 US disclosed
CN-1252068-A 3-piperidyl-4-oxoquinazoline derivatives and pharmaceutical compositions containing the same JAPAN TOBACCO INC (JP) 2000-05-03 CN disclosed
EP-0970954-A1 3-PIPERIDYL-4-OXOQUINAZOLINE DERIVATIVES AND MEDICINCAL COMPOSITIONS CONTAINING THE SAME JAPAN TOBACCO INC. (JP) 2000-01-12 EP disclosed