SCHEMBL7979955

SCHEMBL7979955

Cc1cccc(Cl)c1-c1ncc2c(N)nc3ccc(NCCN(C)C)cc3n12

nearest known ligand 0.54

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
LCK P06239 11/20 0.54
KDR P35968 2/20 0.37
NOS1 P29475 1/20 0.37
NOS2 P35228 1/20 0.37
FGFR1 P11362 1/20 0.36
PDE2A O00408 5/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7979828 0.93 LCK (0.48) LCKKDRNOS1NOS2FGFR1
SCHEMBL7982709 0.93 LCK (0.53) LCKKDRNOS1NOS2FGFR1
SCHEMBL7987029 0.88 LCK (0.45) LCKKDRFGFR1PDE2A
SCHEMBL7983062 0.88 LCK (0.50) LCKKDRFGFR1PDE2A
SCHEMBL7981128 0.87 LCK (0.54) LCKKDRFGFR1
SCHEMBL7982991 0.87 LCK (0.43) LCKKDRFGFR1PDE2A
SCHEMBL7982930 0.86 LCK (0.51) LCKKDRFGFR1PDE2A
SCHEMBL7987537 0.86 LCK (0.42) LCKKDRFGFR1PDE2A
SCHEMBL4038826 0.86 FGFR1 (0.49) LCKKDRFGFR1
SCHEMBL7983214 0.86 LCK (0.51) LCKKDRFGFR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6235740-B1 AUTOIMMUNE DISEASES; ANTIPROLIFERATION AGENTS BRISTOL-MYERS SQUIBB CO. 2001-05-22 US claimed
WO-1999009845-A1 IMIDAZOQUINOXALINE PROTEIN TYROSINE KINASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 1999-03-04 WO claimed
US-6235740-B1 AUTOIMMUNE DISEASES; ANTIPROLIFERATION AGENTS BRISTOL-MYERS SQUIBB CO. 2001-05-22 US disclosed