SCHEMBL7987029

SCHEMBL7987029

CN(C)CCCNc1ccc2nc(N)c3cnc(-c4c(F)cccc4Cl)n3c2c1

nearest known ligand 0.45

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
LCK P06239 4/20 0.45
WEE1 P30291 1/20 0.39
PDE2A O00408 6/20 0.39
FGFR1 P11362 3/20 0.38
KDR P35968 2/20 0.38
MAP4K4 O95819 1/20 0.38
CDK9 P50750 2/20 0.37
PDE10A Q9Y233 1/20 0.36
FLT3 P36888 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7982991 0.97 LCK (0.43) LCKWEE1PDE2AFGFR1KDR
SCHEMBL7987537 0.97 LCK (0.42) LCKWEE1PDE2AFGFR1KDR
SCHEMBL7979828 0.95 LCK (0.48) LCKPDE2AFGFR1KDRPDE10A
SCHEMBL7979955 0.88 LCK (0.54) LCKPDE2AFGFR1KDR
SCHEMBL7981128 0.86 LCK (0.54) LCKWEE1FGFR1KDRMAP4K4
SCHEMBL7983672 0.85 FGFR1 (0.53) LCKFGFR1KDR
SCHEMBL7982930 0.83 LCK (0.51) LCKWEE1PDE2AFGFR1KDR
SCHEMBL7969691 0.83 NPC1 (0.39) LCKPDE2ACDK9PDE10A
SCHEMBL7983214 0.83 LCK (0.51) LCKWEE1FGFR1KDRCDK9
SCHEMBL7980015 0.83 LCK (0.52) LCKPDE2AFGFR1KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6235740-B1 AUTOIMMUNE DISEASES; ANTIPROLIFERATION AGENTS BRISTOL-MYERS SQUIBB CO. 2001-05-22 US claimed
US-6235740-B1 AUTOIMMUNE DISEASES; ANTIPROLIFERATION AGENTS BRISTOL-MYERS SQUIBB CO. 2001-05-22 US disclosed