SCHEMBL7980106

SCHEMBL7980106

COc1ccc(-c2ccc(-c3nc(C4=CC(=S)CC=C4)c(NC(=O)c4ccccc4)o3)c(O)c2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 3/20 0.42
MAPT P10636 8/20 0.41
MEN1 O00255 6/20 0.41
KMT2A Q03164 6/20 0.41
ALDH1A1 P00352 4/20 0.41
KDM4E B2RXH2 3/20 0.41
HPGD P15428 3/20 0.41
POLB P06746 2/20 0.41
HSD17B10 Q99714 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
GAA P10253 1/20 0.41
RAB9A P51151 4/20 0.41
NPC1 O15118 3/20 0.41
TSHR P16473 1/20 0.41
HDAC2 Q92769 1/20 0.40
FLT1 P17948 1/20 0.39
FLT4 P35916 1/20 0.39
ABCG2 Q9UNQ0 1/20 0.38
ADORA3 P0DMS8 2/20 0.38
TP53 P04637 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7746568 0.93 KDR (0.41) KDRMAPTMEN1KMT2AALDH1A1
SCHEMBL7986013 0.91 KDR (0.39) KDRMAPTMEN1KMT2AALDH1A1
SCHEMBL7980279 0.89 KDR (0.47) KDRMAPTMEN1KMT2AALDH1A1
SCHEMBL7969457 0.86 KDR (0.42) KDRMAPTMEN1KMT2AKDM4E
SCHEMBL7986526 0.86 KDR (0.42) KDRMAPTMEN1KMT2AALDH1A1
SCHEMBL7744769 0.85 KDR (0.53) KDRALDH1A1KDM4EPOLBSMN1; SMN2
SCHEMBL7969509 0.85 MCL1 (0.38) KDRMAPTMEN1KMT2AALDH1A1
SCHEMBL7739003 0.84 HPN (0.44) KDRMAPTMEN1KMT2AALDH1A1
SCHEMBL7982878 0.83 MAPT (0.44) KDRMAPTMEN1KMT2AALDH1A1
SCHEMBL7744069 0.80 KDR (0.40) KDRMAPTALDH1A1KDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6228871-B1 THIAZOLE OR OXAZOLE DERIVATIVE TYROSINE KINASE INHIBITORS; ANTICARCINOGENIC AGENTS; AUTOIMMUNE DISEASES; DIABETIC RETINOPATHY MERCK & CO., INC. 2001-05-08 US claimed