SCHEMBL7986013

SCHEMBL7986013

Cc1ccc(-c2ccc(-c3nc(C4=CC(=S)CC=C4)c(NC(=O)c4ccccc4)o3)c(O)c2)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 2/20 0.39
FLT1 P17948 1/20 0.39
FLT4 P35916 1/20 0.39
MAPT P10636 6/20 0.38
KDM4E B2RXH2 7/20 0.37
MEN1 O00255 6/20 0.37
KMT2A Q03164 6/20 0.37
POLB P06746 3/20 0.37
AGPAT2 O15120 1/20 0.37
NPC1 O15118 2/20 0.37
RAB9A P51151 2/20 0.37
HPGD P15428 5/20 0.36
HTT P42858 2/20 0.36
LMNA P02545 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
ALDH1A1 P00352 5/20 0.35
KCNMA1 Q12791 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC2 Q92769 1/20 0.34
HSD17B10 Q99714 3/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7746568 0.95 KDR (0.41) KDRFLT1FLT4MAPTKDM4E
SCHEMBL7980106 0.91 KDR (0.42) KDRFLT1FLT4MAPTKDM4E
SCHEMBL7982717 0.89 KDR (0.44) KDRFLT1FLT4MAPTKDM4E
SCHEMBL7969457 0.89 KDR (0.42) KDRFLT1FLT4MAPTKDM4E
SCHEMBL7986526 0.89 KDR (0.42) KDRFLT1FLT4MAPTKDM4E
SCHEMBL7744769 0.87 KDR (0.53) KDRFLT1FLT4KDM4EPOLB
SCHEMBL7969509 0.87 MCL1 (0.38) KDRFLT1FLT4MAPTKDM4E
SCHEMBL7739003 0.86 HPN (0.44) KDRFLT1FLT4MAPTKDM4E
SCHEMBL7979629 0.82 KDR (0.39) KDRFLT1FLT4MAPTKDM4E
SCHEMBL7744069 0.82 KDR (0.40) KDRFLT1FLT4MAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6228871-B1 THIAZOLE OR OXAZOLE DERIVATIVE TYROSINE KINASE INHIBITORS; ANTICARCINOGENIC AGENTS; AUTOIMMUNE DISEASES; DIABETIC RETINOPATHY MERCK & CO., INC. 2001-05-08 US claimed