SCHEMBL7980768

SCHEMBL7980768

CC(=O)Nc1oc(-c2ccc(-c3ccc(C)cc3)cc2O)nc1C1=CC=CCC1=S

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 7/20 0.45
FLT1 P17948 1/20 0.45
FLT4 P35916 1/20 0.45
NPC1 O15118 3/20 0.36
RAB9A P51151 3/20 0.36
RXFP1 Q9HBX9 1/20 0.36
ADORA3 P0DMS8 3/20 0.34
POLB P06746 3/20 0.33
KMT2A Q03164 3/20 0.33
MEN1 O00255 2/20 0.33
KDM4E B2RXH2 1/20 0.33
AGPAT2 O15120 1/20 0.33
MAPT P10636 3/20 0.32
HSP90AA1 P07900 1/20 0.32
ESR1 P03372 1/20 0.32
GAA P10253 1/20 0.32
TNNI3 P19429 1/20 0.32
TNNT2 P45379 1/20 0.32
TNNC1 P63316 1/20 0.32
ESR2 Q92731 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7744196 0.93 KDR (0.54) KDRFLT1FLT4NPC1RAB9A
SCHEMBL7979629 0.89 KDR (0.39) KDRFLT1FLT4NPC1RAB9A
SCHEMBL7986670 0.88 KDR (0.50) KDRFLT1FLT4NPC1RAB9A
SCHEMBL7744746 0.85 HPN (0.45) KDRFLT1FLT4POLBMAPT
SCHEMBL7744779 0.84 KDR (0.43) KDRFLT1FLT4NPC1RAB9A
SCHEMBL7981618 0.84 KDR (0.44) KDRFLT1FLT4
SCHEMBL7979897 0.81 KDR (0.47) KDRFLT1FLT4NPC1RAB9A
SCHEMBL7982717 0.81 KDR (0.44) KDRFLT1FLT4NPC1RAB9A
SCHEMBL7744056 0.80 HPGD (0.42) KDRFLT1FLT4NPC1RAB9A
SCHEMBL7982878 0.80 MAPT (0.44) KDRFLT1FLT4NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6228871-B1 THIAZOLE OR OXAZOLE DERIVATIVE TYROSINE KINASE INHIBITORS; ANTICARCINOGENIC AGENTS; AUTOIMMUNE DISEASES; DIABETIC RETINOPATHY MERCK & CO., INC. 2001-05-08 US claimed