SCHEMBL7979897

SCHEMBL7979897

CC(=O)Nc1oc(-c2cccc(-c3ccc(-c4ccc5ccccc5c4)cc3)c2O)nc1C1=CC=CCC1=S

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 7/20 0.47
FLT1 P17948 1/20 0.47
FLT4 P35916 1/20 0.47
UTRN P46939 2/20 0.38
ALOX15 P16050 1/20 0.37
NPC1 O15118 3/20 0.33
RAB9A P51151 3/20 0.33
MAP4K4 O95819 1/20 0.33
ROS1 P08922 1/20 0.33
FLT3 P36888 1/20 0.33
MAPK8 P45983 1/20 0.33
GSK3B P49841 1/20 0.33
ITK Q08881 1/20 0.33
DYRK1A Q13627 1/20 0.33
AURKB Q96GD4 1/20 0.33
CLK4 Q9HAZ1 1/20 0.33
HSD17B1 P14061 1/20 0.32
HSD17B2 P37059 1/20 0.32
HDAC4 P56524 1/20 0.32
HDAC2 Q92769 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7744196 0.84 KDR (0.54) KDRFLT1FLT4ALOX15NPC1
SCHEMBL7979682 0.83 KDR (0.46) KDRFLT1FLT4UTRNALOX15
SCHEMBL7980768 0.81 KDR (0.45) KDRFLT1FLT4NPC1RAB9A
SCHEMBL7986670 0.80 KDR (0.50) KDRFLT1FLT4ALOX15NPC1
SCHEMBL7979899 0.79 KDR (0.52) KDRFLT1FLT4UTRNALOX15
SCHEMBL7979692 0.78 KDR (0.54) KDRFLT1FLT4UTRNALOX15
SCHEMBL7982616 0.78 KDR (0.56) KDRFLT1FLT4UTRNALOX15
SCHEMBL7981618 0.78 KDR (0.44) KDRFLT1FLT4ALOX15CLK4
SCHEMBL7744746 0.77 HPN (0.45) KDRFLT1FLT4MAPTTP53
SCHEMBL7744779 0.76 KDR (0.43) KDRFLT1FLT4NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6228871-B1 THIAZOLE OR OXAZOLE DERIVATIVE TYROSINE KINASE INHIBITORS; ANTICARCINOGENIC AGENTS; AUTOIMMUNE DISEASES; DIABETIC RETINOPATHY MERCK & CO., INC. 2001-05-08 US claimed