SCHEMBL7981618

SCHEMBL7981618

CC(=O)Nc1oc(-c2ccc(-c3ccccc3C(F)(F)F)cc2O)nc1C1=CC=CCC1=S

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 7/20 0.44
FLT1 P17948 1/20 0.44
FLT4 P35916 1/20 0.44
CYP1A2 P05177 2/20 0.34
TSHR P16473 2/20 0.34
CNR2 P34972 1/20 0.34
USP2 O75604 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C19 P33261 1/20 0.34
CLK4 Q9HAZ1 1/20 0.34
ATR Q13535 1/20 0.34
ALOX15 P16050 1/20 0.33
PIK3R1 P27986 1/20 0.32
PIK3CA P42336 1/20 0.32
MCHR1 Q99705 1/20 0.32
DHODH Q02127 1/20 0.32
SCN9A Q15858 2/20 0.31
KDM4C Q9H3R0 1/20 0.31
TRPA1 O75762 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7744196 0.87 KDR (0.54) KDRFLT1FLT4TSHRATR
SCHEMBL7986670 0.84 KDR (0.50) KDRFLT1FLT4TSHRATR
SCHEMBL7980768 0.84 KDR (0.45) KDRFLT1FLT4
SCHEMBL7744746 0.80 HPN (0.45) KDRFLT1FLT4ATR
SCHEMBL7744779 0.79 KDR (0.43) KDRFLT1FLT4TSHR
SCHEMBL7979897 0.78 KDR (0.47) KDRFLT1FLT4CLK4ALOX15
SCHEMBL7979629 0.77 KDR (0.39) KDRFLT1FLT4TSHR
SCHEMBL7744056 0.75 HPGD (0.42) KDRFLT1FLT4CYP1A2TSHR
SCHEMBL7987348 0.75 KDR (0.44) KDRFLT1FLT4
SCHEMBL7982878 0.75 MAPT (0.44) KDRFLT1FLT4TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6228871-B1 THIAZOLE OR OXAZOLE DERIVATIVE TYROSINE KINASE INHIBITORS; ANTICARCINOGENIC AGENTS; AUTOIMMUNE DISEASES; DIABETIC RETINOPATHY MERCK & CO., INC. 2001-05-08 US claimed