SCHEMBL7980930

SCHEMBL7980930

C[Si](C)(C)OC1(C#N)CCc2cc(Cl)ccc21

nearest known ligand 0.37

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 2/20 0.37
SRD5A1 P18405 11/20 0.36
ESR1 P03372 5/20 0.34
ESR2 Q92731 5/20 0.34
SRD5A2 P31213 1/20 0.34
KEAP1 Q14145 1/20 0.34
NFE2L2 Q16236 1/20 0.34
KCNA5 P22460 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23891554 0.84 ADRA2A (0.38) ESR1ESR2
SCHEMBL1530577 0.83 BACE1 (0.35) KDM1AESR1ESR2
SCHEMBL9364462 0.83 ADRA2A (0.43) KDM1A
SCHEMBL3900065 0.82 KDM1A (0.43) KDM1AKEAP1NFE2L2
SCHEMBL7973198 0.80 KDM1A (0.36) KDM1A
SCHEMBL17605796 0.76 ALDH1A1 (0.41)
SCHEMBL23997717 0.76 SIGMAR1 (0.32)
SCHEMBL17236222 0.76 KDM4E (0.32)
SCHEMBL11170633 0.76 MAP3K14 (0.39)
SCHEMBL3020640 0.76 KDM1A (0.36) KDM1AESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001045704-A1 INHIBITORS OF PRENYL-PROTEIN TRANSFERASE MERCK & CO., INC. (US) 2001-06-28 WO disclosed