SCHEMBL7981909

SCHEMBL7981909

N#Cc1ccc(C(O)(c2ccc(Cl)cc2)c2cn(C(c3ccccc3)(c3ccccc3)c3ccccc3)cn2)cc1

nearest known ligand 0.38

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ACSS2 Q9NR19 1/20 0.38
CYP19A1 P11511 10/20 0.38
CYP3A4 P08684 1/20 0.38
CYP3A5 P20815 1/20 0.38
RORC P51449 5/20 0.36
MAOA P21397 1/20 0.33
MAOB P27338 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2915674 0.94 CYP3A4 (0.41) ACSS2CYP19A1CYP3A4CYP3A5
SCHEMBL7984249 0.84 S1PR3 (0.38) CYP19A1CYP3A4CYP3A5RORC
SCHEMBL2918068 0.83 CYP19A1 (0.39) ACSS2CYP19A1CYP3A4CYP3A5
SCHEMBL7980280 0.78 FNTA (0.42) CYP19A1RORC
SCHEMBL7984344 0.77 CYP19A1 (0.37) CYP19A1CYP3A4CYP3A5RORC
SCHEMBL5688661 0.73 CYP17A1 (0.44) CYP19A1CYP3A4RORC
SCHEMBL4032019 0.73 ACSS2 (0.38) ACSS2CYP3A4RORC
SCHEMBL5689382 0.72 CYP17A1 (0.43) ACSS2CYP3A4RORC
SCHEMBL914557 0.71 CYP3A4 (0.57) ACSS2CYP19A1CYP3A4CYP3A5MAOA
SCHEMBL2787655 0.71 CYP19A1 (0.36) ACSS2CYP19A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6297239-B1 Inhibitors of prenyl-protein transferase MERCK & CO., INC. 2001-10-02 US disclosed