SCHEMBL7982034

SCHEMBL7982034

CCc1cc(C#Cc2ccc(C3(NCCc4ccccc4)CC3)cc2)ccc1C(=O)O

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HNF4A P41235 1/20 0.39
FFAR1 O14842 6/20 0.38
PTGES O14684 1/20 0.35
ACACB O00763 2/20 0.35
RARA P10276 2/20 0.35
RARB P10826 2/20 0.35
RARG P13631 2/20 0.35
CYP26A1 O43174 1/20 0.35
CYP3A4 P08684 1/20 0.35
CRABP2 P29373 1/20 0.35
FFAR4 Q5NUL3 1/20 0.34
KDM4E B2RXH2 1/20 0.33
ASPH Q12797 1/20 0.33
RIOX2 Q8IUF8 1/20 0.33
KDM8 Q8N371 1/20 0.33
ADRB1 P08588 1/20 0.33
ADRB3 P13945 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7982021 0.89 HNF4A (0.38) HNF4AFFAR1PTGESACACBRARA
SCHEMBL7980637 0.88 RARB (0.36) HNF4APTGESRARARARBRARG
SCHEMBL5737003 0.82 RARB (0.43) FFAR1ACACBRARARARBRARG
SCHEMBL5737932 0.78 KMT2A (0.49) CYP3A4
SCHEMBL7554831 0.78 OPRM1 (0.50) HNF4APTGESRARARARBRARG
SCHEMBL7987895 0.77 HNF4A (0.38) HNF4AFFAR1ACACBRARARARB
SCHEMBL7988083 0.73 RARB (0.38) HNF4AFFAR1RARARARBRARG
SCHEMBL5736570 0.71 RARB (0.46) ACACBRARARARBRARGCYP26A1
SCHEMBL7971273 0.70 RARB (0.36) HNF4AFFAR1RARARARBRARG
SCHEMBL7984179 0.70 RARB (0.36) HNF4AACACBRARARARBRARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6303785-B1 SUBSTITUTED N-CYCLOPROPYLTETRAHYDROISOQUINOLINES ALLERGAN SALES, INC. 2001-10-16 US disclosed