SCHEMBL7971273

SCHEMBL7971273

CCCN(CCC)C1(c2ccc(C#Cc3ccc(C(=O)O)c(CC)c3)cc2)CC1

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
RARB P10826 10/20 0.36
RARG P13631 9/20 0.36
RARA P10276 6/20 0.36
CYP26A1 O43174 1/20 0.36
CYP3A4 P08684 1/20 0.36
CRABP2 P29373 1/20 0.36
HNF4A P41235 1/20 0.35
PTPN11 Q06124 1/20 0.33
PTPRO Q16827 1/20 0.33
RXRA P19793 2/20 0.32
OPRM1 P35372 3/20 0.31
OPRL1 P41146 3/20 0.31
HCAR3 P49019 1/20 0.30
FFAR1 O14842 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5737278 0.83 RARB (0.46) RARBRARGRARACYP26A1CYP3A4
SCHEMBL7554831 0.80 OPRM1 (0.50) RARBRARGRARACYP26A1CYP3A4
SCHEMBL7988083 0.77 RARB (0.38) RARBRARGRARACYP26A1CYP3A4
SCHEMBL7980637 0.77 RARB (0.36) RARBRARGRARACYP26A1CYP3A4
SCHEMBL7984179 0.74 RARB (0.36) RARBRARGRARACYP26A1CYP3A4
SCHEMBL10412862 0.72 GABRP (0.41) HNF4ARXRAFFAR1
SCHEMBL7982021 0.72 HNF4A (0.38) RARBRARGRARACYP26A1CYP3A4
SCHEMBL7987895 0.72 HNF4A (0.38) RARBRARGRARACYP26A1CYP3A4
SCHEMBL7982034 0.70 HNF4A (0.39) RARBRARGRARACYP26A1CYP3A4
SCHEMBL7987639 0.69 HNF4A (0.37) RARBRARGRARAHNF4AFFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6303785-B1 SUBSTITUTED N-CYCLOPROPYLTETRAHYDROISOQUINOLINES ALLERGAN SALES, INC. 2001-10-16 US disclosed