SCHEMBL7988083

SCHEMBL7988083

CCc1cc(C#Cc2ccc(C3(OC)CC3)cc2)ccc1C(=O)O

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
RARB P10826 6/20 0.38
RARG P13631 5/20 0.38
RARA P10276 3/20 0.38
CYP26A1 O43174 1/20 0.38
CYP3A4 P08684 1/20 0.38
CRABP2 P29373 1/20 0.38
HNF4A P41235 1/20 0.37
RXRA P19793 2/20 0.34
NEK2 P51955 1/20 0.33
FFAR1 O14842 3/20 0.33
ALOX5 P09917 1/20 0.33
PTPN11 Q06124 1/20 0.32
PPARG P37231 1/20 0.32
PPARA Q07869 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7984179 0.87 RARB (0.36) RARBRARGRARACYP26A1CYP3A4
SCHEMBL7987895 0.84 HNF4A (0.38) RARBRARGRARACYP26A1CYP3A4
SCHEMBL5737036 0.78 RARB (0.51) RARBRARGRARACYP26A1CYP3A4
SCHEMBL7980637 0.77 RARB (0.36) RARBRARGRARACYP26A1CYP3A4
SCHEMBL7971273 0.77 RARB (0.36) RARBRARGRARACYP26A1CYP3A4
SCHEMBL7980771 0.77 RARB (0.38) RARBRARGRARACYP26A1CYP3A4
SCHEMBL7982021 0.77 HNF4A (0.38) RARBRARGRARACYP26A1CYP3A4
SCHEMBL5736135 0.75 FFAR1 (0.55) FFAR1ALOX5
SCHEMBL10412862 0.75 GABRP (0.41) HNF4ARXRANEK2FFAR1PPARG
SCHEMBL7970709 0.75 RARB (0.39) RARBRARGRARACYP26A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6303785-B1 SUBSTITUTED N-CYCLOPROPYLTETRAHYDROISOQUINOLINES ALLERGAN SALES, INC. 2001-10-16 US disclosed