SCHEMBL7982677

SCHEMBL7982677

Nc1cccn2cc(CCO)nc12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 5/20 0.47
NPC1 O15118 4/20 0.47
RAB9A P51151 4/20 0.47
MAPT P10636 4/20 0.47
DHFR P00374 1/20 0.46
MAPK1 P28482 3/20 0.38
TP53 P04637 1/20 0.38
SIRT5 Q9NXA8 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
HTR2A P28223 1/20 0.37
HTR2C P28335 1/20 0.37
ALDH1A1 P00352 3/20 0.36
LMNA P02545 1/20 0.36
KDM4E B2RXH2 6/20 0.36
TSHR P16473 1/20 0.36
HTT P42858 1/20 0.36
POLB P06746 1/20 0.35
HSD17B10 Q99714 3/20 0.34
HPGD P15428 2/20 0.34
ALDH1A2 O94788 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9226257 0.80 SMN1; SMN2 (0.52) SMN1; SMN2NPC1RAB9AMAPTDHFR
SCHEMBL2489626 0.76 RAB9A (0.49) SMN1; SMN2NPC1RAB9AMAPTDHFR
SCHEMBL7982689 0.72 ALDH1A1 (0.46) SMN1; SMN2NPC1RAB9AMAPTDHFR
SCHEMBL7834962 0.71 PDE10A (0.59) SMN1; SMN2NPC1RAB9AMAPTMAPK1
SCHEMBL2403951 0.70 DHFR (0.48) SMN1; SMN2NPC1RAB9AMAPTDHFR
Hydrochloric Acid SCHEMBL9081198 0.69 DHFR (0.47) SMN1; SMN2NPC1RAB9AMAPTDHFR
Bromide SCHEMBL9099637 0.69 DHFR (0.47) SMN1; SMN2NPC1RAB9AMAPTDHFR
SCHEMBL8373781 0.69 PTGS1 (0.54) SMN1; SMN2NPC1RAB9AMAPTDHFR
SCHEMBL23320338 0.68 MAPK1 (0.40) SMN1; SMN2NPC1RAB9AMAPTMAPK1
SCHEMBL14736747 0.68 NPC1 (0.57) SMN1; SMN2NPC1RAB9AMAPTMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6174877-B1 EXCELLANT BACTERICIDES, ORAL ABSORBABILITY AND STABILITY; IMPROVE THE STABILITY TO RENAL DEHYDROPEPTIDASE I (DHP-I); 2-(2-(N-HETEROCYCLIC-ETHYLTHIO-) DERIVATIVES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-01-16 US disclosed
EP-0876370-A1 CARBAPENEM COMPOUNDS, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1998-11-11 EP disclosed
WO-1997025325-A1 CARBAPENEM COMPOUNDS, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-07-17 WO disclosed