SCHEMBL7982687

SCHEMBL7982687

CCCC(=O)Oc1cn2cccc(N)c2n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHFR P00374 1/20 0.41
MAPT P10636 3/20 0.35
RAB9A P51151 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
NPC1 O15118 1/20 0.35
HTR2A P28223 1/20 0.35
HTR2C P28335 1/20 0.35
KDM4E B2RXH2 2/20 0.34
HSD17B10 Q99714 2/20 0.34
KMT2A Q03164 2/20 0.34
ALDH1A1 P00352 2/20 0.34
MEN1 O00255 1/20 0.34
ALOX15 P16050 1/20 0.34
CASP1 P29466 1/20 0.34
TSPO P30536 1/20 0.33
CA2 P00918 2/20 0.33
MTNR1A P48039 1/20 0.33
MTNR1B P49286 1/20 0.33
BCL9 O00512 1/20 0.33
CTNNB1 P35222 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7980862 0.77 PTGS1 (0.47) MAPTRAB9ASMN1; SMN2NPC1KDM4E
SCHEMBL7986875 0.74 KDM4E (0.53) RAB9ASMN1; SMN2NPC1KDM4EHSD17B10
SCHEMBL7982712 0.74 BCL9 (0.34) MAPTRAB9ASMN1; SMN2NPC1KDM4E
SCHEMBL7982689 0.72 ALDH1A1 (0.46) DHFRMAPTRAB9ASMN1; SMN2NPC1
SCHEMBL118201 0.71 ALDH1A1 (0.56) DHFRMAPTRAB9ASMN1; SMN2NPC1
SCHEMBL7982679 0.70 GAA (0.39) MAPTRAB9ASMN1; SMN2HTR2AHTR2C
SCHEMBL7982993 0.69 KDM4E (0.39) MAPTRAB9AKDM4EKMT2AALDH1A1
SCHEMBL7981083 0.68 HRH4 (0.42) RAB9AKDM4EHSD17B10KMT2AALDH1A1
SCHEMBL9226257 0.68 SMN1; SMN2 (0.52) DHFRMAPTRAB9ASMN1; SMN2NPC1
SCHEMBL8373781 0.67 PTGS1 (0.54) DHFRMAPTRAB9ASMN1; SMN2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6174877-B1 EXCELLANT BACTERICIDES, ORAL ABSORBABILITY AND STABILITY; IMPROVE THE STABILITY TO RENAL DEHYDROPEPTIDASE I (DHP-I); 2-(2-(N-HETEROCYCLIC-ETHYLTHIO-) DERIVATIVES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-01-16 US disclosed
EP-0876370-A1 CARBAPENEM COMPOUNDS, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1998-11-11 EP disclosed
WO-1997025325-A1 CARBAPENEM COMPOUNDS, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-07-17 WO disclosed