SCHEMBL7983280

SCHEMBL7983280

Oc1ccc2c(c1O)C(Cc1ccncc1)c1ccccc1-2

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 10/20 0.39
HTR2A P28223 1/20 0.34
KDM4E B2RXH2 1/20 0.33
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
CYP3A4 P08684 1/20 0.33
BCL2 P10415 1/20 0.33
MAPT P10636 1/20 0.33
HPGD P15428 1/20 0.33
ALOX15 P16050 1/20 0.33
ALOX12 P18054 1/20 0.33
MAOA P21397 1/20 0.33
APEX1 P27695 1/20 0.33
MAPK1 P28482 1/20 0.33
RECQL P46063 1/20 0.33
DAPK1 P53355 1/20 0.33
KMT2A Q03164 1/20 0.33
MCL1 Q07820 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
CYP1B1 Q16678 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7987343 0.88 HTR2A (0.38) HTR2AKDM4EMEN1ALDH1A1CYP3A4
SCHEMBL8111113 0.80 CYP19A1 (0.47) CYP19A1HTR2ACYP3A4MAPTALOX15
SCHEMBL9816167 0.79 HTR2A (0.40) HTR2AKDM4EMEN1ALDH1A1CYP3A4
Hydrochloric Acid SCHEMBL9719344 0.78 CYP19A1 (0.46) CYP19A1HTR2ACYP3A4MAPTALOX15
SCHEMBL7983255 0.76 LOXL2 (0.39) HTR2AKDM4EMEN1ALDH1A1CYP3A4
SCHEMBL7987634 0.74 ADRB2 (0.39) BCL2ALOX15
SCHEMBL9269160 0.73 CYP19A1 (0.41) CYP19A1HTR2ACYP3A4ALOX15MAOA
SCHEMBL9266327 0.73 CYP19A1 (0.41) CYP19A1HTR2ACYP3A4ALOX15MAOA
SCHEMBL30779227 0.73 HTR2A (0.40) HTR2AMEN1ALDH1A1MAPTHPGD
SCHEMBL8840931 0.71 CES2 (0.41) HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6194439-B1 ANTICANCER AGENT PFIZER INC. 2001-02-27 US disclosed
EP-0586608-A1 TRICYCLIC POLYHYDROXYLIC TYROSINE KINASE INHIBITORS PFIZER INC. (US) 1994-03-16 EP disclosed
WO-1992021660-A1 TRICYCLIC POLYHYDROXYLIC TYROSINE KINASE INHIBITORS PFIZER, INC. (US) 1992-12-10 WO disclosed