SCHEMBL7986598

SCHEMBL7986598

Clc1cccc(-c2cncc(-c3cn(CCN4CCOCC4)c4cccc(Cl)c34)c2)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 5/20 0.53
FLT1 P17948 3/20 0.53
FLT4 P35916 3/20 0.53
MAPK13 O15264 1/20 0.43
MAPK12 P53778 1/20 0.43
MAPK11 Q15759 1/20 0.43
MAPK14 Q16539 1/20 0.43
NFATC1 O95644 1/20 0.41
GSK3B P49841 1/20 0.41
DYRK1A Q13627 1/20 0.41
CNR2 P34972 1/20 0.40
KDM4E B2RXH2 2/20 0.39
TSHR P16473 2/20 0.39
MEN1 O00255 1/20 0.39
LMNA P02545 1/20 0.39
MAPT P10636 1/20 0.39
KMT2A Q03164 1/20 0.39
ALDH1A1 P00352 1/20 0.39
POLB P06746 1/20 0.39
PDE4B Q07343 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7986909 0.92 KDR (0.57) KDRFLT1FLT4NFATC1GSK3B
SCHEMBL7990426 0.91 KDR (0.54) KDRFLT1FLT4NFATC1GSK3B
SCHEMBL7548475 0.91 KDR (0.52) KDRFLT1FLT4ALDH1A1GRIN1
SCHEMBL7553606 0.88 KDR (0.49) KDRFLT1FLT4GSK3BTSHR
SCHEMBL7987083 0.87 KDR (0.69) KDRFLT1FLT4MAPK13MAPK12
SCHEMBL7990322 0.86 KDR (0.73) KDRFLT1FLT4NFATC1GSK3B
SCHEMBL7554600 0.85 KDR (0.54) KDRFLT1FLT4MAPK13MAPK12
SCHEMBL7552023 0.85 KDR (0.40) KDRFLT1FLT4TSHRMEN1
SCHEMBL7976802 0.85 KDR (0.59) KDRFLT1FLT4MAPK13MAPK12
SCHEMBL7976928 0.85 KDR (0.59) KDRFLT1FLT4MAPK13MAPK12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6306865-B1 SYNTHASE INHIBITORS AND ANTITUMOR AGENTS GLAXO WELLCOME INC. 2001-10-23 US disclosed
US-6265403-B1 TYROSINE INHIBITORS MERCK & CO., INC. 2001-07-24 US disclosed