SCHEMBL7986664

SCHEMBL7986664

COc1ccc(-c2cncc(-c3cn(C(C)CN(C)C)c4cccc(Cl)c34)c2)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 2/20 0.40
KDR P35968 2/20 0.37
FLT1 P17948 1/20 0.37
FLT4 P35916 1/20 0.37
CYP11B1 P15538 7/20 0.35
CYP11B2 P19099 7/20 0.35
MAP4K4 O95819 1/20 0.35
PDE4B Q07343 1/20 0.35
PDE4D Q08499 1/20 0.35
KMT2A Q03164 1/20 0.33
CYP17A1 P05093 1/20 0.33
CHRNB1 P11230 1/20 0.33
CHRNB2 P17787 1/20 0.33
CHRNB4 P30926 1/20 0.33
CHRNA3 P32297 1/20 0.33
CHRNB3 Q05901 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
ALPL P05186 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7990817 0.92 KDR (0.36) KDRFLT1FLT4CYP11B1CYP11B2
SCHEMBL7986476 0.90 KDR (0.39) KDRFLT1FLT4MAP4K4CHRNB1
SCHEMBL7548486 0.89 KDR (0.41) KDRFLT1FLT4PLA2G4A
SCHEMBL7986898 0.85 KDR (0.38) KDRFLT1FLT4
SCHEMBL7551047 0.85 KDR (0.51) MAOBKDRFLT1FLT4CYP11B1
SCHEMBL7572831 0.85 MAOB (0.39) MAOBKDRCYP11B1CYP11B2MAP4K4
SCHEMBL7550587 0.84 KDR (0.49) KDRFLT1FLT4CYP11B1CYP11B2
SCHEMBL7553622 0.83 KDR (0.55) KDRFLT1FLT4CYP3A4CYP2C9
SCHEMBL7990418 0.82 KDR (0.39) KDRFLT1FLT4CYP11B1CYP11B2
SCHEMBL7549809 0.81 HTR6 (0.43) KDRFLT1FLT4CYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265403-B1 TYROSINE INHIBITORS MERCK & CO., INC. 2001-07-24 US disclosed