SCHEMBL7986901

SCHEMBL7986901

CC(C1CCCNC1)n1cc(-c2cncc(-c3ccsc3)c2)c2ccc(Cl)cc21

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 8/20 0.41
FLT1 P17948 4/20 0.41
FLT4 P35916 4/20 0.41
CHEK1 O14757 4/20 0.36
CDK2 P24941 3/20 0.36
CCNA2 P20248 2/20 0.36
CCNA1 P78396 2/20 0.36
CYP2A6 P11509 3/20 0.36
CCNT1 O60563 1/20 0.35
CCNE1 P24864 1/20 0.35
CDK7 P50613 1/20 0.35
CDK9 P50750 1/20 0.35
CCNH P51946 1/20 0.35
MNAT1 P51948 1/20 0.35
PRKCZ Q05513 1/20 0.34
TDP2 O95551 1/20 0.32
KCNH2 Q12809 1/20 0.32
PDPK1 O15530 1/20 0.32
RPS6KB1 P23443 1/20 0.32
NFATC1 O95644 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7548212 0.93 KDR (0.39) KDRFLT1FLT4CHEK1CDK2
SCHEMBL7987644 0.89 CCNT1 (0.40) CHEK1CDK2CCNT1CCNE1CDK7
SCHEMBL7510914 0.89 KDR (0.51) KDRFLT1FLT4CHEK1CDK2
SCHEMBL7548474 0.88 CDK7 (0.42) CHEK1CDK2CCNA2CCNA1CCNT1
SCHEMBL7986848 0.87 CCNT1 (0.38) CHEK1CDK2CCNT1CCNE1CDK7
SCHEMBL7991016 0.85 CCNT1 (0.37) CHEK1CDK2CCNT1CCNE1CDK7
SCHEMBL7993811 0.84 KDR (0.39) KDRFLT1FLT4CHEK1CDK2
SCHEMBL7993904 0.83 KDR (0.38) KDRFLT1FLT4CHEK1CDK2
SCHEMBL7976003 0.83 PRKCZ (0.40) KDRFLT1FLT4CHEK1CDK2
SCHEMBL7990984 0.83 CCNT1 (0.36) CHEK1CDK2CCNT1CCNE1CDK7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265403-B1 TYROSINE INHIBITORS MERCK & CO., INC. 2001-07-24 US disclosed