SCHEMBL7993904

SCHEMBL7993904

CC(C1CCCNC1)n1cc(-c2cncc(-c3ccsc3)c2)c2cc(C#N)ccc21

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KDR P35968 8/20 0.38
FLT1 P17948 4/20 0.38
FLT4 P35916 4/20 0.38
CYP2A6 P11509 3/20 0.34
KDM1A O60341 3/20 0.34
CHEK1 O14757 3/20 0.34
CCNA2 P20248 2/20 0.34
CDK2 P24941 2/20 0.34
CCNA1 P78396 2/20 0.34
PRKCZ Q05513 1/20 0.33
IDH2 P48735 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7548212 0.88 KDR (0.39) KDRFLT1FLT4CYP2A6CHEK1
SCHEMBL7505916 0.88 CCNT1 (0.38) KDM1ACDK2PRKCZ
SCHEMBL7510914 0.87 KDR (0.51) KDRFLT1FLT4CYP2A6CHEK1
SCHEMBL7976003 0.87 PRKCZ (0.40) KDRFLT1FLT4CYP2A6CHEK1
SCHEMBL7994416 0.87 CCNT1 (0.37) KDM1ACDK2
SCHEMBL7990500 0.85 KDM1A (0.41) KDM1ACHEK1
SCHEMBL7975983 0.85 CCNT1 (0.36) KDM1ACDK2
SCHEMBL7986901 0.83 KDR (0.41) KDRFLT1FLT4CYP2A6CHEK1
SCHEMBL7990463 0.83 CHEK1 (0.39) KDM1ACHEK1
SCHEMBL7994041 0.80 KDR (0.41) KDRFLT1FLT4CYP2A6CHEK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265403-B1 TYROSINE INHIBITORS MERCK & CO., INC. 2001-07-24 US disclosed