SCHEMBL7987263

SCHEMBL7987263

COc1ccc(C(=O)C2CNCCN2CC2(C)Cc3c(C)c(N)c(C)c(C)c3O2)cc1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP1 P03956 3/20 0.34
MMP9 P14780 3/20 0.34
MMP13 P45452 3/20 0.34
MMP3 P08254 1/20 0.34
MMP7 P09237 1/20 0.34
KDM2B Q8NHM5 3/20 0.32
GAA P10253 2/20 0.32
ALDH1A1 P00352 3/20 0.32
LMNA P02545 2/20 0.32
CHRNB2 P17787 2/20 0.31
CHRNB4 P30926 2/20 0.31
CHRNA3 P32297 2/20 0.31
CHRNA7 P36544 2/20 0.31
CHRNA4 P43681 2/20 0.31
POLB P06746 2/20 0.31
KMT2A Q03164 1/20 0.31
UGCG Q16739 1/20 0.31
OPRM1 P35372 1/20 0.31
OPRD1 P41143 1/20 0.31
KDM4E B2RXH2 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8579633 0.65 DRD3 (0.40) GAAALDH1A1LMNAKMT2ASMN1; SMN2
Hydrochloric Acid SCHEMBL6983896 0.64 SIGMAR1 (0.48) GAAALDH1A1LMNAKMT2AKDM4E
SCHEMBL6984000 0.64 LGMN (0.40) GAAALDH1A1KMT2AKDM4EMAPT
SCHEMBL27662026 0.63 MMP1 (0.45) MMP1MMP9MMP13MMP3MMP7
SCHEMBL6981092 0.62 DRD3 (0.34) GAALMNAKMT2AOPRM1MAPT
SCHEMBL21120758 0.60 KDM2B (0.66) KDM2BALDH1A1KDM4E
Hydrochloric Acid SCHEMBL6981668 0.59 SIGMAR1 (0.38) GAAALDH1A1LMNAPOLBKMT2A
SCHEMBL5427255 0.59 MMP1 (0.39) MMP1MMP9MMP13MMP3MMP7
SCHEMBL8719900 0.58 AKT1 (0.33) LMNAKMT2AMAPT
SCHEMBL28109125 0.57 REN (0.47) GAAALDH1A1CHRNB2CHRNB4CHRNA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6172085-B1 CENTRAL NERVOUS SYSTEM AND PSYCHOLOGICAL DISORDERS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-01-09 US disclosed