SCHEMBL7987703

SCHEMBL7987703

O=C(N=C1c2cc(O)c(O)cc2-c2cc(O)c(O)cc21)c1ccc(C(F)(F)F)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.46
CES1 P23141 2/20 0.46
IGFBP3 P17936 1/20 0.42
SRD5A2 P31213 1/20 0.41
GPR6 P46095 1/20 0.40
GSK3B P49841 2/20 0.40
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
PTPN1 P18031 2/20 0.40
CRHBP P24387 1/20 0.40
CRHR2 Q13324 1/20 0.40
LMNA P02545 2/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
MAPT P10636 1/20 0.39
PTGS2 P35354 1/20 0.39
TTR P02766 1/20 0.39
SRC P12931 1/20 0.39
PRKACA P17612 1/20 0.39
PRKACG P22612 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7983607 0.73 HTR3E (0.43) CES2CES1RAB9ALMNAMEN1
SCHEMBL10986357 0.69 CES2 (0.59) CES2CES1SRD5A2GSK3BPTPN1
SCHEMBL6993491 0.66 CES2 (0.55) CES2CES1SRD5A2GSK3BPTPN1
SCHEMBL3294022 0.66 KIF11 (0.60) NQO2
SCHEMBL648641 0.65 SRD5A2 (0.83) CES2CES1SRD5A2GSK3BNPC1
SCHEMBL3172262 0.65 CES2 (1.00) CES2CES1SRD5A2GSK3BPTPN1
SCHEMBL28472299 0.65 CES2 (0.53) CES2CES1SRD5A2GSK3BPTPN1
Hydrochloric Acid SCHEMBL8505964 0.65 CES2 (0.53) CES2CES1SRD5A2GSK3BPTPN1
SCHEMBL23968981 0.64 KIF11 (0.47)
SCHEMBL7983283 0.64 NQO2 (0.54) PTGS2NQO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6194439-B1 ANTICANCER AGENT PFIZER INC. 2001-02-27 US disclosed
EP-0586608-A1 TRICYCLIC POLYHYDROXYLIC TYROSINE KINASE INHIBITORS PFIZER INC. (US) 1994-03-16 EP disclosed
WO-1992021660-A1 TRICYCLIC POLYHYDROXYLIC TYROSINE KINASE INHIBITORS PFIZER, INC. (US) 1992-12-10 WO disclosed