SCHEMBL7983283

SCHEMBL7983283

Oc1cc2c(cc1O)-c1cc(O)c(O)cc1C2=Cc1ccc(C(F)(F)F)cc1

nearest known ligand 0.54

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
NQO2 P16083 2/20 0.54
PTGS1 P23219 5/20 0.47
PTGS2 P35354 2/20 0.46
RXRA P19793 1/20 0.42
CYP1A2 P05177 2/20 0.41
AHR P35869 1/20 0.40
PIM1 P11309 1/20 0.39
PIM2 Q9P1W9 1/20 0.39
KIF11 P52732 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7987352 0.79 LCK (0.47) NQO2PTGS1PTGS2CYP1A2PIM1
SCHEMBL9372014 0.78 NFE2L2 (0.44) NQO2PTGS1RXRA
SCHEMBL7980865 0.75 LCK (0.46)
SCHEMBL8072577 0.73 MAOA (0.49) CYP1A2AHRPIM1PIM2
SCHEMBL30692069 0.71 CES2 (0.58) CYP1A2
SCHEMBL29153446 0.71 CES2 (0.58) CYP1A2
SCHEMBL29153447 0.71 CES2 (0.58) CYP1A2
SCHEMBL4264937 0.70 NQO2 (1.00) NQO2PTGS1PTGS2CYP1A2AHR
SCHEMBL4264940 0.70 NQO2 (1.00) NQO2PTGS1PTGS2CYP1A2AHR
SCHEMBL4157456 0.70 CYP19A1 (0.46) CYP1A2PIM1PIM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6194439-B1 ANTICANCER AGENT PFIZER INC. 2001-02-27 US disclosed
EP-0586608-A1 TRICYCLIC POLYHYDROXYLIC TYROSINE KINASE INHIBITORS PFIZER INC. (US) 1994-03-16 EP disclosed
WO-1992021660-A1 TRICYCLIC POLYHYDROXYLIC TYROSINE KINASE INHIBITORS PFIZER, INC. (US) 1992-12-10 WO disclosed