SCHEMBL7990800

SCHEMBL7990800

O=c1cc(-c2ccncc2)[nH]c(NCCc2ccc(Cl)cc2Cl)n1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR84 Q9NQS5 1/20 0.49
TAAR1 Q96RJ0 1/20 0.46
ROCK2 O75116 2/20 0.39
ROCK1 Q13464 1/20 0.39
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
DPP4 P27487 1/20 0.38
CASP1 P29466 1/20 0.38
PDE9A O76083 1/20 0.37
KMT2A Q03164 2/20 0.37
GCGR P47871 3/20 0.37
MAPK14 Q16539 2/20 0.37
CNR1 P21554 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
DAO P14920 1/20 0.36
LMNA P02545 1/20 0.36
TSHR P16473 1/20 0.36
MAPK1 P28482 1/20 0.36
GSK3A P49840 1/20 0.36
GSK3B P49841 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1841756 0.82 GPR84 (0.49) GPR84TAAR1ROCK2ROCK1CYP3A4
SCHEMBL7992854 0.81 GPR84 (0.41) GPR84ROCK2ROCK1KMT2AGCGR
SCHEMBL5382412 0.79 CYP3A4 (0.41) GPR84TAAR1ROCK2ROCK1CYP3A4
SCHEMBL7993027 0.77 CA1 (0.40) TAAR1ROCK2CYP3A4KMT2AGCGR
SCHEMBL7978450 0.77 GPR84 (0.44) GPR84ROCK2GCGRMAPK14LMNA
SCHEMBL7993029 0.76 GPR84 (0.50) GPR84KMT2AGSK3B
SCHEMBL5390245 0.76 PRKCA (0.43) GPR84ROCK2KMT2AGSK3BHPGD
SCHEMBL7978256 0.74 HTR2A (0.43) GPR84KMT2ALMNAHPGD
SCHEMBL5375269 0.72 CDC7 (0.43) LMNAGSK3BHPGD
SCHEMBL7992535 0.72 PTGDR (0.50) CYP3A4CYP2C9KMT2ALMNATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001070727-A1 2-(ARYLALKYLAMINO)PYRIMIDONE DERIVATIVES AND 2-(HETEROARYLALKYLAMINO)PYRIMIDONE DERIVATIVES SANOFI-SYNTHELABO (FR) 2001-09-27 WO claimed