SCHEMBL7991609

SCHEMBL7991609

COc1cccc(C(=O)C2=NCCc3cc(OCc4ccccc4)ccc32)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 5/20 0.49
MRGPRX4 Q96LA9 3/20 0.49
SRD5A2 P31213 1/20 0.49
NR4A2 P43354 1/20 0.48
SMPD1 P17405 2/20 0.47
VNN1 O95497 1/20 0.46
MAOA P21397 3/20 0.46
RAB9A P51151 2/20 0.45
TP53 P04637 1/20 0.45
PKM P14618 1/20 0.45
NFKB1 P19838 1/20 0.45
NFKB2 Q00653 1/20 0.45
RELA Q04206 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
RXFP1 Q9HBX9 1/20 0.45
HPD P32754 1/20 0.43
NPC1 O15118 1/20 0.43
POLB P06746 1/20 0.43
GFER P55789 1/20 0.43
PAX8 Q06710 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7988818 0.91 MAOB (0.48) MAOBMRGPRX4SRD5A2VNN1MAOA
SCHEMBL7994780 0.90 MAOB (0.53) MAOBMRGPRX4SRD5A2NR4A2SMPD1
SCHEMBL7989235 0.87 ACHE (0.48) MAOBSMPD1MAOARAB9ATP53
SCHEMBL7991437 0.87 KDM4E (0.48) MAOBMRGPRX4SRD5A2VNN1
SCHEMBL7991147 0.83 MAOB (0.47) MAOBMAOARAB9ATP53SMN1; SMN2
SCHEMBL7994703 0.80 KDM4E (0.45) MAOBMRGPRX4SRD5A2NR4A2RAB9A
SCHEMBL7977331 0.78 KDM4E (0.49) SMPD1RAB9ASMN1; SMN2NPC1
SCHEMBL7991229 0.78 KDM4E (0.49) RAB9ANPC1
SCHEMBL7992415 0.78 KDM4E (0.51) MRGPRX4SMPD1RAB9ASMN1; SMN2NPC1
SCHEMBL7988142 0.78 KDM4E (0.53) MRGPRX4SMPD1RAB9APKMSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001055117-A1 NOVEL ISOQUINOLINE DERIVATIVES, PREPARATION METHOD AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM LES LABORATOIRES SERVIER (FR) 2001-08-02 WO disclosed