SCHEMBL7993257

SCHEMBL7993257

NS(=O)(=O)c1cc(Cl)c(Cl)c(Cl)c1

nearest known ligand 0.75

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 15/20 0.75
CA1 P00915 14/20 0.75
CA9 Q16790 11/20 0.75
CA7 P43166 4/20 0.75
CA4 P22748 4/20 0.75
CA12 O43570 3/20 0.75
CA6 P23280 3/20 0.75
CA5A P35218 3/20 0.75
CA14 Q9ULX7 3/20 0.75
CA5B Q9Y2D0 3/20 0.75
CA13 Q8N1Q1 2/20 0.75
LMNA P02545 1/20 0.75
CYP2C9 P11712 1/20 0.75
APEX1 P27695 2/20 0.61
POLB P06746 1/20 0.61
TDP1 Q9NUW8 1/20 0.61
L3MBTL1 Q9Y468 1/20 0.61
CA3 P07451 2/20 0.48
CYP2C19 P33261 1/20 0.46
VCAM1 P19320 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Dichlorphenamide SCHEMBL112376 0.86 CA1 (1.00) CA2CA1CA9CA7CA4
Dichlorphenamide SCHEMBL29355725 0.86 CA1 (1.00) CA2CA1CA9CA7CA4
Dichlorphenamide SCHEMBL7034594 0.84 CA1 (0.96) CA2CA1CA9CA7CA4
Dichlorphenamide SCHEMBL7040074 0.84 CA1 (0.96) CA2CA1CA9CA7CA4
Dichlorphenamide SCHEMBL4312398 0.84 CA1 (0.96) CA2CA1CA9CA7CA4
SCHEMBL3781532 0.82 CA1 (1.00) CA2CA1CA9CA7CA4
SCHEMBL5564627 0.80 CA1 (0.64) CA2CA1CA9CA7CA4
SCHEMBL2535790 0.80 CA2 (0.56) CA2CA1CA9CA7CA4
SCHEMBL4333676 0.78 CA1 (0.48) CA2CA1CA9CA7CA4
SCHEMBL11929253 0.77 CA1 (0.68) CA2CA1CA9CA7CA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6281240-B1 CYSTIC FIBROSIS ELI LILLY AND COMPANY 2001-08-28 US disclosed
WO-1998044799-A1 DIARYLSULFONYLUREAS FOR USE IN TREATING SECRETORY DIARRHEA ELI LILLY AND COMPANY (US) 1998-10-15 WO disclosed
EP-0550157-B1 Antitumor compositions and methods of treatment LILLY CO ELI (US) 1997-07-23 EP disclosed
US-5354778-A N-Phenyl-N'-substituted phenylsulfonylureas ELI LILLY AND COMPANY (US) 1994-10-11 US disclosed
EP-0606723-A1 Imidazolidin-2-one derivatives and their use as antitumor agents ELI LILLY AND COMPANY (US) 1994-07-20 EP disclosed
US-5270329-A 1-arylsulfonyl-imidazolidin-2-one derivatives ELI LILLY AND COMPANY (US) 1993-12-14 US disclosed
US-5234955-A N-phenyl-N*-substituted phenylsulfonylureas ELI LILLY AND COMPANY (US) 1993-08-10 US disclosed
EP-0550157-A1 Antitumor compositions and methods of treatment ELI LILLY AND COMPANY (US) 1993-07-07 EP disclosed