SCHEMBL7995157

SCHEMBL7995157

CC(C)c1ccc(CN(C)C(=O)N=C(N)NOS(C)(=O)=O)cc1S(C)(=O)=O

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SLC9A1 P19634 3/20 0.46
SLC9A2 Q9UBY0 1/20 0.45
HSP90AA1 P07900 7/20 0.33
HDAC3 O15379 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC7 Q8WUI4 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP3A5 P20815 1/20 0.32
CYP3A7 P24462 1/20 0.32
CYP2C19 P33261 1/20 0.32
CYP3A43 Q9HB55 1/20 0.32
CTSD P07339 1/20 0.31
MAPK8 P45983 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8004814 0.81 CTSD (0.36) CTSD
SCHEMBL8097928 0.80 SLC9A1 (0.53) SLC9A1SLC9A2HSP90AA1HDAC3HDAC1
SCHEMBL4355373 0.77 SLC9A1 (0.72) SLC9A1SLC9A2
SCHEMBL27524440 0.75 SLC9A1 (0.40) SLC9A1SLC9A2HSP90AA1HDAC3HDAC1
SCHEMBL8007047 0.70 SLC9A1 (0.60) SLC9A1SLC9A2
Hydrochloric Acid SCHEMBL8004970 0.69 SLC9A1 (0.58) SLC9A1SLC9A2
Water SCHEMBL8088760 0.69 SLC9A1 (0.50) SLC9A1SLC9A2
SCHEMBL8007941 0.66 SLC9A1 (0.49) SLC9A1SLC9A2
SCHEMBL7995153 0.66 SLC9A1 (0.49) SLC9A1SLC9A2MAPK8
SCHEMBL8097379 0.65 SLC9A1 (0.50) SLC9A1SLC9A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0748795-B1 Substituted benzyloxycarbonyl guanidines as Na+/H+ exchange inhibitors, process for their preparation, their use as medicinal or diagnostic agents as well as medicament containing them HOECHST AG (DE) 2000-08-23 EP claimed
US-6022899-A EFFECTIVE INHIBITORS OF THE CELLULAR SODIUM PROTON ANTIPORTER HOECHST AKTIENGESELLSCHAFT (DE) 2000-02-08 US claimed
US-6022899-A EFFECTIVE INHIBITORS OF THE CELLULAR SODIUM PROTON ANTIPORTER HOECHST AKTIENGESELLSCHAFT (DE) 2000-02-08 US disclosed
US-5753710-A INHIBITORS OF THE CELLULAR SODIUM PROTON ANTIPORTER HOECHST AKTIENGESELLSCHAFT (DE) 1998-05-19 US disclosed