SCHEMBL7995963

SCHEMBL7995963

CCc1c(-c2ccc(OC)cc2)nn(-c2ccccc2)c1-c1ccc(OC)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 1/20 0.52
PTGS2 P35354 1/20 0.52
CCNA2 P20248 1/20 0.50
CDK2 P24941 1/20 0.50
RAB9A P51151 5/20 0.48
KDM4E B2RXH2 4/20 0.48
SMN1; SMN2 Q16637 3/20 0.48
HTT P42858 3/20 0.48
ALDH1A1 P00352 6/20 0.48
KMT2A Q03164 5/20 0.48
LMNA P02545 4/20 0.48
MEN1 O00255 4/20 0.48
NPC1 O15118 3/20 0.48
NPSR1 Q6W5P4 3/20 0.48
MAPT P10636 2/20 0.48
TP53 P04637 2/20 0.48
GMNN O75496 1/20 0.48
USP2 O75604 1/20 0.48
ESR1 P03372 1/20 0.48
CYP1A2 P05177 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8009492 0.93 TP53 (0.55) PTGS1PTGS2CCNA2CDK2KDM4E
SCHEMBL11248919 0.84 PTGDR2 (0.50) PTGS1PTGS2CCNA2CDK2RAB9A
SCHEMBL5217314 0.83 ESR1 (0.68) PTGS1PTGS2RAB9AKDM4ESMN1; SMN2
SCHEMBL11245609 0.81 ALDH1A1 (0.48) CCNA2CDK2KDM4EHTTALDH1A1
SCHEMBL23403668 0.80 RPA1 (0.47) RAB9AKDM4ESMN1; SMN2HTTALDH1A1
SCHEMBL11251973 0.80 RPA1 (0.50) PTGS2CCNA2CDK2RAB9AKDM4E
SCHEMBL5218437 0.79 CDK2 (0.45) PTGS1PTGS2CCNA2CDK2RAB9A
SCHEMBL8008424 0.79 L3MBTL1 (0.52) RAB9AKDM4ESMN1; SMN2HTTALDH1A1
SCHEMBL21121386 0.78 ESR1 (0.64) KDM4EALDH1A1MAPTTP53ESR1
SCHEMBL11733429 0.77 PTGS2 (0.51) PTGS1PTGS2CCNA2CDK2RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000019994-A9 ESTROGEN RECEPTOR LIGANDS UNIV ILLINOIS (US) 2000-08-31 WO disclosed
WO-2000019994-A1 ESTROGEN RECEPTOR LIGANDS BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS (US) 2000-04-13 WO disclosed