SCHEMBL7996541

SCHEMBL7996541

Fc1cc(-c2c3cccccc-3nc2-c2cccc(Cl)c2)ccn1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 7/20 0.46
ADORA2A P29274 6/20 0.46
NQO2 P16083 2/20 0.46
PIM1 P11309 1/20 0.43
TDO2 P48775 1/20 0.41
MAPK13 O15264 1/20 0.41
RAF1 P04049 1/20 0.41
MAPK12 P53778 1/20 0.41
MAPK11 Q15759 1/20 0.41
MAPK14 Q16539 1/20 0.41
ADORA1 P30542 3/20 0.41
KMO O15229 1/20 0.41
IDO1 P14902 1/20 0.41
NPC1 O15118 1/20 0.40
MITF O75030 1/20 0.40
TP53 P04637 1/20 0.40
MAPT P10636 1/20 0.40
PKM P14618 1/20 0.40
TSHR P16473 1/20 0.40
GRM5 P41594 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7997046 0.84 MAPK11 (0.54) ADORA2BADORA2APIM1MAPK13RAF1
SCHEMBL7997004 0.83 MAPK14 (0.48) ADORA2BADORA2ANQO2MAPK13MAPK12
SCHEMBL8000428 0.82 MAPK14 (0.54) ADORA2ATDO2MAPK13RAF1MAPK12
SCHEMBL30930875 0.71 NUDT1 (0.40) ADORA2BADORA2ANQO2MAPK13MAPK12
SCHEMBL30930949 0.70 NUDT1 (0.42) PIM1MAPK14KMO
SCHEMBL15637672 0.68 RORB (0.55) ADORA2BADORA2APIM1TDO2MAPK13
SCHEMBL31472663 0.68 NOTUM (0.48) ADORA2BIDO1MAPTGRM5
SCHEMBL21333215 0.68 NOTUM (0.48) ADORA2BIDO1MAPTGRM5
SCHEMBL7993062 0.68 MAPK14 (0.50) ADORA2AMAPK13RAF1MAPK12MAPK11
SCHEMBL15637561 0.68 GRM5 (0.52) ADORA2APIM1TDO2ADORA1IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001057018-A1 AZAAZULENE INHIBITORS OF P38 MAP KINASE AND TNF-ALPHA ABBOTT LABORATORIES (US) 2001-08-09 WO claimed
WO-2001057018-A1 AZAAZULENE INHIBITORS OF P38 MAP KINASE AND TNF-ALPHA ABBOTT LABORATORIES (US) 2001-08-09 WO disclosed