SCHEMBL7999929

SCHEMBL7999929

N=C(N)c1ccc(CN2CCN(C(=O)c3ccc(-c4ccccc4)cc3)CC2=O)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 1/20 0.52
DPP4 P27487 1/20 0.50
ITGB3 P05106 1/20 0.47
ITGA2B P08514 1/20 0.47
TSHR P16473 3/20 0.46
LMNA P02545 2/20 0.46
ALDH1A1 P00352 2/20 0.46
NPSR1 Q6W5P4 1/20 0.46
CYP46A1 Q9Y6A2 1/20 0.46
POLB P06746 2/20 0.45
MAPK1 P28482 2/20 0.45
HPGD P15428 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.44
WDR5 P61964 1/20 0.44
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
SLC6A7 Q99884 1/20 0.44
F10 P00742 2/20 0.43
F2 P00734 1/20 0.43
PRSS1 P07477 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7987038 0.89 F10 (0.54) HRH3DPP4LMNAALDH1A1CYP46A1
SCHEMBL7986762 0.85 F10 (0.55) HRH3DPP4ITGB3ITGA2BWDR5
SCHEMBL7996357 0.85 NPC1 (0.54) HRH3ITGB3ITGA2BTSHRLMNA
SCHEMBL7074519 0.82 KDM4E (0.61) TSHRLMNAALDH1A1POLBMAPK1
Trifluoroacetic Acid SCHEMBL7997619 0.82 PRSS1 (0.52) F10F2PRSS1
SCHEMBL7996082 0.81 GPR119 (0.42) HRH3ITGB3ITGA2BLMNACYP46A1
SCHEMBL7986862 0.81 F10 (0.57) TSHRALDH1A1SMN1; SMN2WDR5F10
SCHEMBL4387744 0.81 F2 (0.48) HRH3DPP4ITGB3ITGA2BNPSR1
SCHEMBL7069417 0.80 HPGD (0.68) TSHRLMNAALDH1A1NPSR1POLB
SCHEMBL7997768 0.79 NPC1 (0.49) HRH3TSHRLMNAHPGDF10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000008005-A2 PIPERAZINONE DERIVATIVES MERCK PATENT GMBH (DE) 2000-02-17 WO disclosed