SCHEMBL8000244

SCHEMBL8000244

Cc1ccc(C(=S)Cl)cn1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.52
HDAC6 Q9UBN7 1/20 0.52
KDM4E B2RXH2 2/20 0.42
ADRA2A P08913 2/20 0.39
ADRA2B P18089 2/20 0.39
ADRA2C P18825 2/20 0.39
DGAT1 O75907 1/20 0.39
KMT2A Q03164 3/20 0.38
NAPRT Q6XQN6 1/20 0.38
KCNQ3 O43525 1/20 0.36
KCNQ2 O43526 1/20 0.36
MAPT P10636 1/20 0.36
PRKAB2 O43741 1/20 0.36
PRKAG1 P54619 1/20 0.36
PRKAA2 P54646 1/20 0.36
PRKAA1 Q13131 1/20 0.36
PRKAG3 Q9UGI9 1/20 0.36
PRKAG2 Q9UGJ0 1/20 0.36
PRKAB1 Q9Y478 1/20 0.36
RAB9A P51151 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7948362 0.82 HDAC1 (0.52) HDAC1HDAC6KDM4EADRA2AADRA2B
SCHEMBL1436032 0.80 HDAC1 (0.50) HDAC1HDAC6KDM4EADRA2AADRA2B
SCHEMBL11344489 0.80 HDAC1 (0.50) HDAC1HDAC6KDM4EADRA2AADRA2B
SCHEMBL600144 0.80 HDAC1 (0.60) HDAC1HDAC6KDM4EKMT2ANAPRT
Hydrochloric Acid SCHEMBL3891479 0.78 HDAC1 (0.58) HDAC1HDAC6KDM4EADRA2AADRA2B
SCHEMBL4491812 0.77 HDAC1 (0.47) HDAC1HDAC6KDM4EADRA2AADRA2B
SCHEMBL4491815 0.77 HDAC1 (0.47) HDAC1HDAC6KDM4EADRA2AADRA2B
SCHEMBL4400941 0.74 HDAC1 (0.64) HDAC1HDAC6KDM4EKMT2AKCNQ3
Potassium Ion SCHEMBL7741543 0.74 HDAC1 (0.58) HDAC1HDAC6KDM4EKMT2AKCNQ3
SCHEMBL3394733 0.74 HDAC1 (0.58) HDAC1HDAC6KDM4EKMT2AKCNQ3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6294536-B1 CONTROL OF PROTOZOA AND REDUCTION IN THE INCIDENCE OF ASSOCIATED DISEASES AND DEATH AND CONSEQUENT IMPROVEMENT IN RETARDED GROWTH AND GENERAL CONDITION AND PREVENTING DECREASE GROWTH AND GENERAL CONDITION TAKEDA SCHERING-PLOUGH ANIMAL HEALTH K.K. (JP) 2001-09-25 US disclosed
WO-1999011634-A1 TRIAZINE DERIVATIVES, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1999-03-11 WO disclosed
EP-0163855-B1 NITROMETHYLENE DERIVATIVES, INTERMEDIATES, AND PROCESS FOR THEIR PREPARATION AS INSECTICIDES NIHON TOKUSHU NOYAKU SEIZO K.K. (JP) 1989-06-21 EP disclosed
US-4812571-A NITROMETHYLENE COMPOUNDS NIHON TOKUSHU NOYAKU SEIZO K.K. (JP) 1989-03-14 US disclosed
US-4774247-A Nitromethylene derivative insecticides NIHON TOKUSHU NOYAKU SEIZO K.K. (JP) 1988-09-27 US disclosed
US-4678795-A 1-pyridylmethyl-2-nitromethylene-1,3-diazacycloalkane insecticides NIHON TOKUSHU NOYAKU SEIZO K.K. (JP) 1987-07-07 US disclosed
EP-0163855-A1 Nitromethylene derivatives, intermediates, and process for their preparation as insecticides NIHON TOKUSHU NOYAKU SEIZO K.K. (JP) 1985-12-11 EP disclosed