SCHEMBL8001598

SCHEMBL8001598

COc1cc2[nH]cc(CC(C)O)c2cc1F

nearest known ligand 0.54

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 3/20 0.54
HTR2B P41595 3/20 0.52
MTNR1A P48039 3/20 0.49
MTNR1B P49286 2/20 0.47
HTR2A P28223 3/20 0.47
HTR2C P28335 3/20 0.47
GPR84 Q9NQS5 2/20 0.45
HTR1D P28221 1/20 0.43
HTR1B P28222 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
NFKB1 P19838 1/20 0.43
CYP2C19 P33261 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL735049 0.81 HTR1A (0.63) HTR1AHTR2BMTNR1AMTNR1BHTR2A
SCHEMBL14527148 0.81 HTR1A (0.63) HTR1AHTR2BMTNR1AHTR2AHTR2C
SCHEMBL7997808 0.75 HTR2A (0.62) HTR1AHTR2BMTNR1AMTNR1BHTR2A
SCHEMBL1196112 0.75 HTR1A (0.75) HTR1AHTR2BMTNR1AMTNR1BHTR2A
SCHEMBL699832 0.75 HTR2A (0.73) HTR1AHTR2AHTR2CGPR84
SCHEMBL7995785 0.74 HTR2B (0.60) HTR1AHTR2BMTNR1AMTNR1BHTR2A
SCHEMBL1196782 0.74 HTR2B (0.61) HTR1AHTR2BMTNR1AMTNR1BHTR2A
SCHEMBL1196780 0.74 HTR2B (0.61) HTR1AHTR2BMTNR1AMTNR1BHTR2A
SCHEMBL2534666 0.74 HTR1A (0.72) HTR1AHTR2BMTNR1AMTNR1BHTR2A
SCHEMBL23259357 0.73 GPR84 (0.65) HTR1AHTR2BHTR2AHTR2CGPR84

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001040183-A1 1-AMINOALKYL-1H-INDOLES FOR TREATING GLAUCOMA ALCON UNIVERSAL LTD. (CH) 2001-06-07 WO disclosed