SCHEMBL8002230

SCHEMBL8002230

Cc1cccc(Cl)c1Cc1cc(-n2nc(-c3cccnc3)nc2C#N)ccc1N

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.35
F2 P00734 1/20 0.35
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
HTT P42858 3/20 0.34
ALDH1A1 P00352 3/20 0.34
HSD17B10 Q99714 2/20 0.34
CHRNB2 P17787 2/20 0.34
CHRNA5 P30532 2/20 0.34
CHRNA4 P43681 2/20 0.34
KDM4E B2RXH2 2/20 0.34
TSHR P16473 1/20 0.34
MAPK1 P28482 1/20 0.34
MAPT P10636 3/20 0.33
KLK7 P49862 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
KCNA5 P22460 1/20 0.33
KCNH2 Q12809 1/20 0.33
CA12 O43570 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7627296 0.81 MAPT (0.36) GAAMEN1KMT2AHTTALDH1A1
SCHEMBL7996172 0.75 CYP11B1 (0.34) F2HSD17B10CHRNB2CHRNA5CHRNA4
SCHEMBL7634848 0.75 MAPT (0.38) F2KMT2AALDH1A1HSD17B10CHRNB2
SCHEMBL7638011 0.71 MAPT (0.45) GAAMEN1KMT2AHTTALDH1A1
SCHEMBL8002213 0.67 CYP11B1 (0.37) F2HTTALDH1A1HSD17B10MAPK1
SCHEMBL7243590 0.66 PTGS2 (0.39) GAAMEN1KMT2AHTTALDH1A1
SCHEMBL7243090 0.66 EPHX2 (0.42) GAAMEN1KMT2AHTTALDH1A1
SCHEMBL7244506 0.58 PTGS2 (0.42) MEN1KMT2AALDH1A1KDM4ENPC1
SCHEMBL7243350 0.58 ALDH1A1 (0.46) MEN1KMT2AALDH1A1HSD17B10KDM4E
SCHEMBL9901553 0.57 ALDH1A1 (0.50) GAAMEN1KMT2AHTTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001072740-A1 SUBSTITUTED 1-(4-AMINOPHENYL) TRIAZOLES AND THEIR USE AS ANTI-INFLAMMATORY AGENTS BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2001-10-04 WO claimed