SCHEMBL8003633

SCHEMBL8003633

C1CNCCSCCN1.[Cu]

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HIF1A Q16665 1/20 0.46
MAPT P10636 1/20 0.46
PDE4A P27815 1/20 0.46
KDR P35968 1/20 0.46
CXCR4 P61073 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
KDM4E B2RXH2 1/20 0.32
GAA P10253 1/20 0.32
CYP2C9 P11712 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1781384 0.96
SCHEMBL8935918 0.96 HIF1A (0.50) HIF1AMAPTPDE4AKDRCXCR4
Piperazine SCHEMBL1063977 0.96 HIF1A (0.50) HIF1AMAPTPDE4AKDRCXCR4
Hydrochloric Acid SCHEMBL7744897 0.92 HIF1A (0.46) HIF1AMAPTPDE4AKDRCXCR4
Bromide SCHEMBL7745419 0.92 HIF1A (0.46) HIF1AMAPTPDE4AKDRCXCR4
Thiomorpholine SCHEMBL145846 0.92
Thiomorpholine SCHEMBL93637 0.92 HIF1A (0.42) HIF1AMAPTPDE4AKDRCXCR4
Thiomorpholine SCHEMBL2273 0.92
SCHEMBL9873225 0.92 HIF1A (0.42) HIF1AMAPTPDE4AKDRCXCR4
Thiomorpholine SCHEMBL253450 0.88

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000010007-A9 DEVICES AND METHODS FOR ANALYSIS OF NON-IONIC SOLUTES CALIFORNIA INST OF TECHN (US) 2000-07-06 WO claimed
US-6063637-A SENSING MATERIAL OF METAL COMPLEXES HAVING AT LEAST TWO COORDINATION SITES FOR BINDING TARGET AND A DETECTOR FOR MEASURING THE PROTONS OR HYDROXIDE IONS RELEASED FROM THE SENSING MATERIAL WHEN ANALYTE IS BOUND CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2000-05-16 US claimed
WO-2000010007-A2 DEVICES AND METHODS FOR ANALYSIS OF NON-IONIC SOLUTES CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2000-02-24 WO claimed
WO-2000010007-A9 DEVICES AND METHODS FOR ANALYSIS OF NON-IONIC SOLUTES CALIFORNIA INST OF TECHN (US) 2000-07-06 WO disclosed
US-6063637-A SENSING MATERIAL OF METAL COMPLEXES HAVING AT LEAST TWO COORDINATION SITES FOR BINDING TARGET AND A DETECTOR FOR MEASURING THE PROTONS OR HYDROXIDE IONS RELEASED FROM THE SENSING MATERIAL WHEN ANALYTE IS BOUND CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2000-05-16 US disclosed
WO-2000010007-A2 DEVICES AND METHODS FOR ANALYSIS OF NON-IONIC SOLUTES CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2000-02-24 WO disclosed