SCHEMBL8004014

SCHEMBL8004014

CC(CCNC1=C(C(=N)C(F)(F)F)CCCC1)C(=O)Nc1cccnc1

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 2/20 0.41
HTT P42858 2/20 0.39
PKM P14618 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
ALDH1A1 P00352 3/20 0.38
CYP3A4 P08684 1/20 0.38
ALOX15 P16050 1/20 0.37
FFAR2 O15552 1/20 0.37
NOTUM Q6P988 1/20 0.37
SMN1; SMN2 Q16637 2/20 0.36
HTR2C P28335 2/20 0.36
HTR2A P28223 1/20 0.36
HTR2B P41595 1/20 0.36
NPC1 O15118 1/20 0.36
LMNA P02545 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8000762 0.88 MME (0.39) RAB9AALDH1A1CYP3A4SMN1; SMN2NPC1
SCHEMBL8004256 0.82 HDAC3 (0.47) PKML3MBTL1NOTUMSMN1; SMN2LMNA
SCHEMBL24767438 0.70 HSD17B10 (0.59) RAB9AHTTPKMALOX15FFAR2
SCHEMBL2435089 0.67 RAB9A (0.60) RAB9AHTTPKMALOX15FFAR2
SCHEMBL21210988 0.66 LMNA (0.64) RAB9AHTTALOX15NPC1LMNA
SCHEMBL12952768 0.65 HDAC3 (0.46) ALDH1A1LMNANPSR1KMT2A
Benzene SCHEMBL7286102 0.65 HTT (0.59) RAB9AHTTPKML3MBTL1ALDH1A1
SCHEMBL18439983 0.64 RAB9A (0.61) RAB9AHTTPKMALOX15FFAR2
SCHEMBL1911526 0.64 HTT (0.67) RAB9AHTTPKMALDH1A1ALOX15
SCHEMBL14032665 0.64 RAB9A (0.64) RAB9AHTTPKMALOX15FFAR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009119088-A1 HETEROCYCLIC COMPOUND 武田薬品工業株式会社 (JP) 2009-10-01 WO disclosed