SCHEMBL8004746

SCHEMBL8004746

COC(=O)c1ccc2c(c1)CCC(c1ccnn1C1CC1)=N2

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.38
TRPA1 O75762 1/20 0.37
BRD4 O60885 1/20 0.36
ALDH1A1 P00352 5/20 0.35
ATM Q13315 2/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
SRD5A1 P18405 1/20 0.35
SRD5A2 P31213 1/20 0.35
PDK1 Q15118 1/20 0.35
PDK2 Q15119 1/20 0.35
PDK3 Q15120 1/20 0.35
PDK4 Q16654 1/20 0.35
KDM4E B2RXH2 4/20 0.35
HPGD P15428 2/20 0.35
GAA P10253 1/20 0.35
TSHR P16473 1/20 0.35
CASP1 P29466 1/20 0.35
CASP7 P55210 1/20 0.35
HSD17B10 Q99714 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16383671 0.73 TRPA1 (0.49) KMT2ATRPA1ALDH1A1ATMSMN1; SMN2
SCHEMBL1963320 0.72 ALOX15 (0.46) KMT2ABRD4ALDH1A1ATMSMN1; SMN2
SCHEMBL19354867 0.71 TRPA1 (0.48) KMT2ATRPA1ALDH1A1ATMSMN1; SMN2
SCHEMBL22039158 0.68 NR3C2 (0.45) KMT2AALDH1A1HPGDTSHRHSD17B10
SCHEMBL17437902 0.67 F2 (0.46) KMT2ABRD4ALDH1A1ATMSMN1; SMN2
SCHEMBL30040346 0.66 HTR1A (0.50) KMT2AALDH1A1ATMSMN1; SMN2NPSR1
SCHEMBL904780 0.66 CYP11B1 (0.47) KMT2AALDH1A1ATMSMN1; SMN2NPSR1
SCHEMBL9644030 0.64 CA1 (0.55) KMT2ATRPA1ALDH1A1ATMSMN1; SMN2
SCHEMBL22672759 0.64 ALDH1A1 (0.47) KMT2ABRD4ALDH1A1ATMSMN1; SMN2
SCHEMBL28062182 0.64 TRPA1 (0.54) KMT2ATRPA1ALDH1A1ATMSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009151991-A1 PYRAZOLE DERIVATIVES USEFUL AS INHIBITORS OF FAAH MERCK & CO., INC. (US) 2009-12-17 WO disclosed