SCHEMBL8004815

SCHEMBL8004815

CC(=CCC(C)N)c1cccc(N)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
F2 P00734 1/20 0.40
PLG P00747 1/20 0.40
PRSS1 P07477 1/20 0.40
PRSS2 P07478 1/20 0.40
PRSS3 P35030 1/20 0.40
PBRM1 Q86U86 1/20 0.39
MEN1 O00255 1/20 0.38
GAA P10253 1/20 0.38
RAB9A P51151 1/20 0.38
KMT2A Q03164 1/20 0.38
ADRB2 P07550 2/20 0.37
ADRB1 P08588 2/20 0.37
ADRB3 P13945 2/20 0.37
NPC1 O15118 1/20 0.37
MITF O75030 1/20 0.37
LMNA P02545 1/20 0.37
POLB P06746 1/20 0.37
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
NOS1 P29475 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9723648 0.81 HTR2A (0.47) HTR2AMAOA
SCHEMBL7519261 0.80 TAAR1 (0.50) PRSS1PRSS2PRSS3RAB9ANPC1
SCHEMBL8867767 0.78 PBRM1 (0.46) F2PLGPRSS1PRSS2PRSS3
SCHEMBL8867994 0.78 PBRM1 (0.46) F2PLGPRSS1PRSS2PRSS3
SCHEMBL7549113 0.77 ALDH1A1 (0.42) F2PLGPRSS1PRSS2PRSS3
SCHEMBL6251422 0.73 MEN1 (0.40) F2PLGPRSS1PRSS2PRSS3
SCHEMBL5199056 0.73 TBXAS1 (0.51) GAALMNAKDM4EALDH1A1CYP3A4
SCHEMBL6251424 0.73 MEN1 (0.40) F2PLGPRSS1PRSS2PRSS3
SCHEMBL7519872 0.72 TP53 (0.37) PRSS1PRSS2PRSS3MEN1RAB9A
SCHEMBL7067559 0.70 HDAC1 (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1042274-A1 PHARMACEUTICAL COMPOSITIONS AND METHODS FOR USE R.J. REYNOLDS TOBACCO COMPANY (US) 2000-10-11 EP claimed
WO-2000023418-A1 PHARMACEUTICAL COMPOSITIONS AND METHODS FOR USE R.J. REYNOLDS TOBACCO COMPANY (US) 2000-04-27 WO claimed
EP-1042274-A1 PHARMACEUTICAL COMPOSITIONS AND METHODS FOR USE R.J. REYNOLDS TOBACCO COMPANY (US) 2000-10-11 EP disclosed
WO-2000023418-A1 PHARMACEUTICAL COMPOSITIONS AND METHODS FOR USE R.J. REYNOLDS TOBACCO COMPANY (US) 2000-04-27 WO disclosed