SCHEMBL8005869

SCHEMBL8005869

CC(=O)c1ccc(CO)c(C)c1N

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.38
PDCD1 Q15116 1/20 0.35
CD274 Q9NZQ7 1/20 0.35
HSD17B1 P14061 1/20 0.35
PDE10A Q9Y233 2/20 0.34
TP53 P04637 1/20 0.34
HSD17B10 Q99714 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.33
MAPT P10636 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
KDM4E B2RXH2 2/20 0.33
ALDH1A1 P00352 1/20 0.33
HPGD P15428 1/20 0.33
METAP2 P50579 1/20 0.32
IKBKB O14920 1/20 0.32
BRD4 O60885 1/20 0.32
GAA P10253 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8008960 0.81 PKM (0.36) PKMHSD17B1KDM4EALDH1A1HPGD
SCHEMBL8280627 0.81 MAPT (0.46) PKMPDCD1CD274HSD17B1SMN1; SMN2
SCHEMBL9890969 0.78 POLB (0.38) TP53HSD17B10SMN1; SMN2MAPTCYP2C9
SCHEMBL1954506 0.76 MAPT (0.43) PKMHSD17B10SMN1; SMN2MAPTCYP2C9
SCHEMBL27668976 0.76 GABRP (0.46) HSD17B10MAPTTDP1KDM4EALDH1A1
SCHEMBL2211047 0.75 POLB (0.50) PDCD1CD274PDE10AHSD17B10SMN1; SMN2
SCHEMBL24507277 0.74 CES2 (0.38) SMN1; SMN2BRD4TSHR
SCHEMBL30560060 0.74 CES2 (0.38) SMN1; SMN2BRD4TSHR
SCHEMBL28700454 0.74 CYP3A4 (0.41) PKMHSD17B1TP53HSD17B10SMN1; SMN2
SCHEMBL10751483 0.73 HSD17B1 (0.42) HSD17B1ALDH1A1HPGDTSHRGABRP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009099596-A2 MACROCYCLIC SERINE PROTEASE INHIBITORS IDENIX PHARAMACEUTICALS, INC. (US) 2009-08-13 WO disclosed