SCHEMBL8006264

SCHEMBL8006264

COC(=O)c1ccc(Oc2ccc3c(c2)COB3)nc1C(=O)OC

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 10/20 0.44
L3MBTL1 Q9Y468 1/20 0.37
ALDH1A1 P00352 2/20 0.34
GPR119 Q8TDV5 2/20 0.34
LMNA P02545 1/20 0.33
TSHR P16473 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
PPARG P37231 2/20 0.33
MAPT P10636 1/20 0.33
GAA P10253 1/20 0.33
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7862584 0.80 PDE4B (0.57) PDE4B
SCHEMBL29541597 0.78 L3MBTL1 (0.46) PDE4BL3MBTL1ALDH1A1LMNATSHR
SCHEMBL2531010 0.77 PDE4B (0.71) PDE4B
SCHEMBL8012386 0.73 PDE4B (0.34) PDE4BALDH1A1
SCHEMBL2531014 0.72 PDE4B (0.68) PDE4B
SCHEMBL3094829 0.70 HRH3 (0.60)
SCHEMBL2529483 0.70 L3MBTL1 (0.39) PDE4BL3MBTL1ALDH1A1GPR119LMNA
SCHEMBL14748429 0.70 PTGS2 (0.43) PDE4BL3MBTL1ALDH1A1GAA
SCHEMBL7902874 0.68 POLB (0.51) L3MBTL1ALDH1A1LMNATSHRNPSR1
SCHEMBL14748452 0.68 P2RX3 (0.35) PDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009111676-A2 BORON-CONTAINING SMALL MOLECULES AS ANTI-INFLAMMATORY AGENTS ANACOR PHARMACEUTICALS, INC (US) 2009-09-11 WO disclosed