Fumaric Acid

Fumaric Acid

SCHEMBL8006607

C=CCc1ccccc1C=C.O=C(O)C=CC(=O)O

nearest known ligand 0.50

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ATP4AATP4BAXLBTKCACNA1CCACNA1DCACNA1FCACNA1SCCR5CHRM2CHRM3CPT1BCPT2DPP4DRD1DRD2EGFRERBB2ERBB4FLT3HRH1HRH3HTR1AHTR2AHTR2BHTR2CHTR4JAK1JAK2JAK3KCNH2KMT2AMAP2K1MAP2K2MEN1MLNRMPLMTORPPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PLK4PPARGRENS1PR1SLC6A2SLC6A3SLC6A4SMOTYK2atpAatpBatpCatpDatpEatpFatpFHatpGpol

The experimentally established mechanism targets of Fumaric Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A known ✓ Q03164 3/20 0.40
MEN1 known ✓ O00255 2/20 0.40
PTGER3 P43115 7/20 0.50
PTGER2 P43116 7/20 0.50
PTGER4 P35408 5/20 0.50
PTGER1 P34995 2/20 0.43
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
NFKB1 P19838 1/20 0.41
CA4 P22748 1/20 0.41
GABRA1 P14867 1/20 0.41
GABRB2 P47870 1/20 0.41
KDM4E B2RXH2 4/20 0.40
SMN1; SMN2 Q16637 3/20 0.40
LMNA P02545 2/20 0.40
MAPT P10636 2/20 0.40
HTT P42858 2/20 0.40
ALOX12 P18054 1/20 0.40
AKR1C3 P42330 1/20 0.40
AKR1C2 P52895 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28185004 0.86 PTGER3 (0.58) PTGER3PTGER2PTGER4PTGER1CA1
SCHEMBL1717109 0.86 PTGER3 (0.67) PTGER3PTGER2PTGER4PTGER1CA1
SCHEMBL30679 0.85 GABRA1 (0.47) NFKB1GABRA1GABRB2KDM4EKMT2A
Methane SCHEMBL28621463 0.83 GABRA1 (0.45) NFKB1GABRA1GABRB2KDM4EKMT2A
Charcoal, Activated SCHEMBL9723291 0.83 GABRA1 (0.45) NFKB1GABRA1GABRB2KDM4EKMT2A
Phenol SCHEMBL27962166 0.82 GABRA1 (0.47) CA1CA2CA4GABRA1GABRB2
Sulfuric Acid SCHEMBL4875624 0.82 POLB (0.45) NFKB1GABRA1GABRB2KDM4ESMN1; SMN2
Maleic Acid SCHEMBL11627287 0.81 CA1 (0.52) PTGER3PTGER2PTGER4CA1CA2
Fumaric Acid SCHEMBL11627288 0.81 CA1 (0.52) PTGER3PTGER2PTGER4CA1CA2
2-Allylphenol SCHEMBL11378333 0.81 AKR1B1 (0.50) PTGER3PTGER2PTGER4CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0665468-B1 Staining inhibitor for photopolymerizable compositions containing a tetrazole MACDERMID IMAGING TECHNOLOGY (US) 2000-04-19 EP disclosed
EP-0665468-A1 Staining inhibitor for photopolymerizable compositions containing a tetrazole HERCULES INCORPORATED (US) 1995-08-02 EP disclosed