SCHEMBL8006987

SCHEMBL8006987

CCc1c(-c2cccc(O)c2)ccc2c1C(=O)NC2=O

nearest known ligand 0.48

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
TDP2 O95551 3/20 0.48
BRAF P15056 2/20 0.48
WEE1 P30291 13/20 0.46
CHEK1 O14757 9/20 0.46
ESR1 P03372 1/20 0.42
ESR2 Q92731 1/20 0.42
USP7 Q93009 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8006796 0.81 CHEK1 (0.51) WEE1CHEK1
SCHEMBL28709463 0.81 TDP2 (0.64) TDP2BRAFWEE1CHEK1
SCHEMBL29652041 0.81 TDP2 (0.64) TDP2BRAFWEE1CHEK1
SCHEMBL8000252 0.80 MAPT (0.48) CHEK1
SCHEMBL10911536 0.72 GSK3B (0.41) WEE1CHEK1
SCHEMBL8757366 0.70 WEE1 (0.50) TDP2BRAFWEE1CHEK1
SCHEMBL9980565 0.70 KDM4E (0.43) WEE1CHEK1
SCHEMBL8690765 0.70 WEE1 (0.50) WEE1CHEK1
SCHEMBL27494083 0.69 PARP1 (0.42) WEE1CHEK1
SCHEMBL27678098 0.69 KDM4E (0.39) WEE1CHEK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000021910-A2 1,2-DISUBSTITUTED CYCLOPROPANES ORTHO-MCNEIL PHARMACEUTICAL, INC. (US) 2000-04-20 WO disclosed