SCHEMBL8000252

SCHEMBL8000252

CCOc1cccc(-c2ccc3c(c2CC)C(=O)NC3=O)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.48
GAA P10253 2/20 0.48
KDM4E B2RXH2 1/20 0.48
THRB P10828 1/20 0.48
TDP1 Q9NUW8 1/20 0.48
CASP3 P42574 1/20 0.44
PTGS2 P35354 1/20 0.42
RXRA P19793 1/20 0.42
RXRB P28702 1/20 0.42
SMN1; SMN2 Q16637 2/20 0.41
TP53 P04637 2/20 0.41
BRD4 O60885 1/20 0.40
BRD2 P25440 1/20 0.40
CREBBP Q92793 1/20 0.40
FGFR1 P11362 2/20 0.39
PDGFRB P09619 1/20 0.39
KDR P35968 1/20 0.39
FABP3 P05413 1/20 0.39
FABP4 P15090 1/20 0.39
FABP5 Q01469 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8006796 0.88 CHEK1 (0.51) GAACASP3BRD4MEN1KMT2A
SCHEMBL8006987 0.80 TDP2 (0.48) CHEK1
SCHEMBL7886526 0.71 CASP3 (0.41) MAPTGAAKDM4ETHRBTDP1
SCHEMBL7886522 0.71 CHRM2 (0.44) MAPTGAAKDM4ETHRBTDP1
SCHEMBL11411139 0.71 MAOA (0.61) MAPTCASP3SMN1; SMN2MEN1KMT2A
SCHEMBL9260410 0.70 RXRA (0.66) MAPTGAAKDM4ETHRBTDP1
SCHEMBL29426410 0.70 RXRA (0.66) MAPTGAAKDM4ETHRBTDP1
SCHEMBL10911536 0.69 GSK3B (0.41) GAAKDM4ECASP3CHEK1HSD17B10
SCHEMBL7399139 0.68 DDB1 (0.46) MAPTGAAKDM4ETHRBTDP1
SCHEMBL29012837 0.68 RXRA (0.64) MAPTGAAKDM4ETHRBTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000021910-A2 1,2-DISUBSTITUTED CYCLOPROPANES ORTHO-MCNEIL PHARMACEUTICAL, INC. (US) 2000-04-20 WO disclosed